Compile Data Set for Download or QSAR
Report error Found 94 Enz. Inhib. hit(s) with all data for entry = 50013290
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060465((Z)-7-[(1S,2R,3R,4R)-3-(4-Phenylethynyl-benzenesul...)
Affinity DataIC50: 8.5nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128694((+) 7-{3-[2-(4-Methoxy-phenyl)-1H-indole-6-sulfony...)
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128711((+) 7-{3-[2-(4-Hydroxy-phenyl)-1H-indole-6-sulfony...)
Affinity DataIC50: 18nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128721(7-[3-(Dibenzofuran-2-sulfonylamino)-bicyclo[2.2.1]...)
Affinity DataIC50: 19nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128693((+) 7-[3-(Dibenzofuran-3-sulfonylamino)-bicyclo[2....)
Affinity DataIC50: 22nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128725((+) 7-[3-(9H-Carbazole-3-sulfonylamino)-bicyclo[2....)
Affinity DataIC50: 22nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128725((+) 7-[3-(9H-Carbazole-3-sulfonylamino)-bicyclo[2....)
Affinity DataIC50: 22nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060447((Z)-7-[(1S,2R,3R,4R)-3-(2-Methoxy-dibenzofuran-3-s...)
Affinity DataIC50: 24nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128711((+) 7-{3-[2-(4-Hydroxy-phenyl)-1H-indole-6-sulfony...)
Affinity DataIC50: 25nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060463((Z)-7-[(1R,2R,6S,7R)-3-(4-Phenylazo-benzenesulfony...)
Affinity DataIC50: 25nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128712(Dibenzofuran-2-sulfonic acid [3-(7-methanesulfonyl...)
Affinity DataIC50: 32nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128703((+) 7-[3-(2-Ethoxy-dibenzofuran-3-sulfonylamino)-b...)
Affinity DataIC50: 32nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128731(7-[3-(2-Methoxy-dibenzofuran-3-sulfonylamino)-bicy...)
Affinity DataIC50: 33nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128707((+) 7-[3-(8-Methoxy-dibenzofuran-2-sulfonylamino)-...)
Affinity DataIC50: 34nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128703((+) 7-[3-(2-Ethoxy-dibenzofuran-3-sulfonylamino)-b...)
Affinity DataIC50: 34nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128701((+) 7-[3-(7-Dimethylamino-dibenzofuran-2-sulfonyla...)
Affinity DataIC50: 36nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128712(Dibenzofuran-2-sulfonic acid [3-(7-methanesulfonyl...)
Affinity DataIC50: 42nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128694((+) 7-{3-[2-(4-Methoxy-phenyl)-1H-indole-6-sulfony...)
Affinity DataIC50: 45nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060448((Z)-7-[(1S,2R,3R,4R)-3-(2-Phenyl-1H-indole-6-sulfo...)
Affinity DataIC50: 47nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060447((Z)-7-[(1S,2R,3R,4R)-3-(2-Methoxy-dibenzofuran-3-s...)
Affinity DataIC50: 52nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128709(7-[3-(2-Methoxy-dibenzofuran-3-sulfonylamino)-bicy...)
Affinity DataIC50: 57nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060451((Z)-7-[(1S,2R,3R,4R)-3-(7-Nitro-dibenzofuran-2-sul...)
Affinity DataIC50: 57nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128724((+) 7-{3-[4-(1-Phenyl-1H-tetrazol-5-yl)-benzenesul...)
Affinity DataIC50: 62nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128729((+) 7-[3-(Dibenzothiophene-2-sulfonylamino)-bicycl...)
Affinity DataIC50: 64nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060461((Z)-7-[(1S,2R,3R,4R)-3-(Dibenzofuran-2-sulfonylami...)
Affinity DataIC50: 70nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060448((Z)-7-[(1S,2R,3R,4R)-3-(2-Phenyl-1H-indole-6-sulfo...)
Affinity DataIC50: 71nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128702((+) 7-[3-(4-Phenylcarbamoyl-benzenesulfonylamino)-...)
Affinity DataIC50: 86nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128699((+) (E) 7-[3-(5-Styryl-thiophene-2-sulfonylamino)-...)
Affinity DataIC50: 90nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128713((+)E 7-[3-(4-Styryl-benzenesulfonylamino)-bicyclo[...)
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128699((+) (E) 7-[3-(5-Styryl-thiophene-2-sulfonylamino)-...)
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128698((+) 7-[3-(4-Benzoylamino-benzenesulfonylamino)-bic...)
Affinity DataIC50: 120nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128704(7-[3-(Dibenzofuran-2-sulfonylamino)-bicyclo[2.2.1]...)
Affinity DataIC50: 120nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128718((+) 7-[3-(2,4,6-Trimethyl-benzenesulfonylamino)-bi...)
Affinity DataIC50: 130nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060461((Z)-7-[(1S,2R,3R,4R)-3-(Dibenzofuran-2-sulfonylami...)
Affinity DataIC50: 130nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128727((+) 7-[3-(4-Phenylamino-benzenesulfonylamino)-bicy...)
Affinity DataIC50: 160nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128693((+) 7-[3-(Dibenzofuran-3-sulfonylamino)-bicyclo[2....)
Affinity DataIC50: 160nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128701((+) 7-[3-(7-Dimethylamino-dibenzofuran-2-sulfonyla...)
Affinity DataIC50: 170nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128713((+)E 7-[3-(4-Styryl-benzenesulfonylamino)-bicyclo[...)
Affinity DataIC50: 180nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128730((+) 7-[3-(2-Hydroxy-dibenzofuran-3-sulfonylamino)-...)
Affinity DataIC50: 180nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50409703(CHEMBL2114171)
Affinity DataIC50: 180nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128729((+) 7-[3-(Dibenzothiophene-2-sulfonylamino)-bicycl...)
Affinity DataIC50: 180nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128728(7-[3-(Dibenzofuran-2-sulfonylamino)-bicyclo[2.2.1]...)
Affinity DataIC50: 180nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128723((+) 7-[3-(1-Methyl-2-phenyl-1H-indole-6-sulfonylam...)
Affinity DataIC50: 190nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128705((+) 7-{3-[4-(1H-Indol-2-yl)-benzenesulfonylamino]-...)
Affinity DataIC50: 190nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128730((+) 7-[3-(2-Hydroxy-dibenzofuran-3-sulfonylamino)-...)
Affinity DataIC50: 190nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128695((+) 7-[3-([2,2']Bithiophenyl-5-sulfonylamino)-bicy...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128700((+) 7-[3-(4'-Methoxy-biphenyl-4-sulfonylamino)-bic...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128716((+) 7-[3-(8-Hydroxy-dibenzofuran-2-sulfonylamino)-...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50409703(CHEMBL2114171)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060465((Z)-7-[(1S,2R,3R,4R)-3-(4-Phenylethynyl-benzenesul...)
Affinity DataIC50: 210nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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