Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50048552
LigandPNGBDBM50220988(CHEMBL544766)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50220984(CHEMBL554636)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM14775(3-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-4-...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50220985(CHEMBL553502)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50220989(CHEMBL542299)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50220990(CHEMBL556179)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50074898(2-[4-(3-Hydroxymethyl-6,7-dimethoxy-naphthalen-1-y...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50074901(2-[4-(2,3-Bis-hydroxymethyl-6,7-dimethoxy-naphthal...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM14775(3-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-4-...)
Affinity DataKi:  0.850nMAssay Description:Inhibition of rolipram binding to phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50220991(CHEMBL539265)
Affinity DataIC50: 1nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50220990(CHEMBL556179)
Affinity DataKi:  1.40nMAssay Description:Inhibition of rolipram binding to phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50220984(CHEMBL554636)
Affinity DataKi:  1.40nMAssay Description:Inhibition of rolipram binding to phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50220985(CHEMBL553502)
Affinity DataKi:  1.5nMAssay Description:Inhibition of rolipram binding to phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50220988(CHEMBL544766)
Affinity DataKi:  1.70nMAssay Description:Inhibition of rolipram binding to phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50220989(CHEMBL542299)
Affinity DataKi:  1.80nMAssay Description:Inhibition of rolipram binding to phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50220986(CHEMBL542650)
Affinity DataIC50: 2nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50074898(2-[4-(3-Hydroxymethyl-6,7-dimethoxy-naphthalen-1-y...)
Affinity DataKi:  3nMAssay Description:Inhibition of rolipram binding to phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50220992(CHEMBL545700)
Affinity DataIC50: 3nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50220986(CHEMBL542650)
Affinity DataKi:  3.10nMAssay Description:Inhibition of rolipram binding to phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50074901(2-[4-(2,3-Bis-hydroxymethyl-6,7-dimethoxy-naphthal...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of rolipram binding to phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM14361(Adeo | 4-(3-cyclopentyloxy-4-methoxy-phenyl)pyrrol...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of rolipram binding to phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50220992(CHEMBL545700)
Affinity DataKi:  5.40nMAssay Description:Inhibition of rolipram binding to phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50220991(CHEMBL539265)
Affinity DataKi:  6.5nMAssay Description:Inhibition of rolipram binding to phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50220987(CHEMBL553278)
Affinity DataIC50: 70nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50220987(CHEMBL553278)
Affinity DataKi:  120nMAssay Description:Inhibition of rolipram binding to phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMed
LigandPNGBDBM14361(Adeo | 4-(3-cyclopentyloxy-4-methoxy-phenyl)pyrrol...)
Affinity DataIC50: 500nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)