Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50003645
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474313(CHEMBL122698)
Affinity DataIC50: 510nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474311(Clinafloxacin)
Affinity DataIC50: 546nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474311(Clinafloxacin)
Affinity DataIC50: 2.73E+3nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474312(CHEMBL120948)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474318(CHEMBL123246)
Affinity DataIC50: 4.26E+3nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474310(CHEMBL121176)
Affinity DataIC50: 4.61E+3nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM21690(Ciprinol | 1-cyclopropyl-6-fluoro-4-oxo-7-(piperaz...)
Affinity DataIC50: 4.82E+3nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474316(CHEMBL331987)
Affinity DataIC50: 7.93E+3nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474312(CHEMBL120948)
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474315(CHEMBL421101)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 2-beta(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474309(CHEMBL331076)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition effect on Escherichia coli Wild Type DNA gyrase Supercoiling activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474317(CHEMBL122691)
Affinity DataIC50: 8.84E+3nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474316(CHEMBL331987)
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474318(CHEMBL123246)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474319(CHEMBL420897)
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474313(CHEMBL122698)
Affinity DataIC50: 3.32E+4nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474315(CHEMBL421101)
Affinity DataIC50: 3.37E+4nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474317(CHEMBL122691)
Affinity DataIC50: 3.59E+4nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474319(CHEMBL420897)
Affinity DataIC50: 3.63E+4nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474314(CHEMBL420884)
Affinity DataIC50: 6.94E+4nMAssay Description:Inhibition of Wild Type DNA gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 2-beta(Human)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474309(CHEMBL331076)
Affinity DataIC50: 7.15E+4nMAssay Description:Inhibition of Escherichia coli Quinolone resistant gyrase Supercoiling activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474314(CHEMBL420884)
Affinity DataIC50: 2.72E+5nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50474310(CHEMBL121176)
Affinity DataIC50: 2.94E+5nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM21690(Ciprinol | 1-cyclopropyl-6-fluoro-4-oxo-7-(piperaz...)
Affinity DataIC50: 3.07E+5nMAssay Description:Inhibition of Quinolone resistant gyrase Supercoiling Activity in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed