Report error Found 155 Enz. Inhib. hit(s) with all data for entry = 50013575
Affinity DataKi: 0.330nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Binding affinity of compound towards human Dopamine receptor D4 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.520nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.560nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.640nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.680nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.730nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.740nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.75nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.920nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Effective concentration for Dopamine receptor D3 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.28nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.31nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.48nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.14nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Effective concentration for Dopamine receptor D3 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 2.85nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.96nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Effective concentration for Dopamine receptor D3 was determined in monkeysMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Binding affinity for human dopamine receptor D2 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Binding affinity for human dopamine receptor D2 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.99nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair












































