Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50013582
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of Src protein tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132153((2,4-Dichloro-5-methoxy-phenyl)-[7-methoxy-8-(2-me...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of Src protein tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132160((2,4-Dichloro-5-methoxy-phenyl)-(7,8-dimethoxy-4a,...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of Src protein tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM4492(CHEMBL101917 | 4-[(2,4-dichlorophenyl)amino]-6,7-d...)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of Src protein tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132158((2,4-Dichloro-5-methoxy-phenyl)-[8-methoxy-7-(2-me...)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of Src protein tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132153((2,4-Dichloro-5-methoxy-phenyl)-[7-methoxy-8-(2-me...)
Affinity DataIC50: 28nMAssay Description:Inhibition of Src protein tyrosine kinase dependent cellular proliferationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM4525(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6,7-dimeth...)
Affinity DataIC50: 30nMAssay Description:Inhibition of Src protein tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Src protein tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132154((2,4-Dichloro-phenyl)-[7-methoxy-8-(2-methoxy-etho...)
Affinity DataIC50: 120nMAssay Description:Inhibition of Src protein tyrosine kinase dependent cellular proliferationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132154((2,4-Dichloro-phenyl)-[7-methoxy-8-(2-methoxy-etho...)
Affinity DataIC50: 120nMAssay Description:Inhibition of Src protein tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132158((2,4-Dichloro-5-methoxy-phenyl)-[8-methoxy-7-(2-me...)
Affinity DataIC50: 140nMAssay Description:Inhibition of Src protein tyrosine kinase dependent cellular proliferationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132160((2,4-Dichloro-5-methoxy-phenyl)-(7,8-dimethoxy-4a,...)
Affinity DataIC50: 190nMAssay Description:Inhibition of Src protein tyrosine kinase dependent cellular proliferationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Fyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 410nMAssay Description:Inhibition of Fyn dependent cellular proliferation of rat 2 fibroblast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132155(7,8-Dimethoxy-5,10-dihydro-1H-pyrimido[4,5-b]quino...)
Affinity DataIC50: 500nMAssay Description:Inhibition of Src protein tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Fyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132153((2,4-Dichloro-5-methoxy-phenyl)-[7-methoxy-8-(2-me...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Fyn dependent cellular proliferation of rat 2 fibroblast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132156((2,4-Dichloro-5-methoxy-phenyl)-(7,8-dimethoxy-pyr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Src protein tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132159((2,4-Dichloro-5-methoxy-phenyl)-[7-methoxy-8-(2-me...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Src protein tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132156((2,4-Dichloro-5-methoxy-phenyl)-(7,8-dimethoxy-pyr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Src protein tyrosine kinase dependent cellular proliferationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132157(7,8-Dimethoxy-3H-pyrimido[4,5-b]quinolin-4-one | 7...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of Src protein tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed