Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 2187
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Morphochem

LigandPNGBDBM17871(1,2,4-triazole derivative. | (1S)-1-[5-(benzylsulf...)
Affinity DataIC50: 43.7nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Morphochem

LigandPNGBDBM17870(1,2,4-triazole derivative. | 5-(benzylsulfanyl)-4H...)
Affinity DataIC50: 599nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Morphochem

LigandPNGBDBM17872(1,2,4-triazole derivative. | 3-(benzylsulfanyl)-4-...)
Affinity DataIC50: 1.00E+5nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2007
Entry Details Article
PubMed