Compile Data Set for Download or QSAR
Report error Found 63 Enz. Inhib. hit(s) with all data for entry = 50013631
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132679(Methyl-((2S,3S)-3-naphthalen-2-yl-bicyclo[2.2.1]he...)
Affinity DataIC50: 9nMAssay Description:In vitro ability of compound to inhibit 5-HT re-uptake of radiolabeled [3H]-tritium transmitter into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132686(Dimethyl-((2S,3S)-3-naphthalen-2-yl-bicyclo[2.2.1]...)
Affinity DataIC50: 9nMAssay Description:In vitro ability of compound to inhibit 5-HT re-uptake of radiolabeled [3H]-tritium transmitter into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132685(Dimethyl-(3-naphthalen-2-yl-bicyclo[2.2.1]hept-2-y...)
Affinity DataIC50: 10nMAssay Description:In vitro ability of compound to inhibit 5-HT re-uptake of radiolabeled [3H]-tritium transmitter into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132677(Dimethyl-((2R,3R)-3-naphthalen-2-yl-bicyclo[2.2.1]...)
Affinity DataIC50: 20nMAssay Description:In vitro ability of compound to inhibit 5-HT re-uptake of radiolabeled [3H]-tritium transmitter into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50026952(CHEMBL322067 | [(2R,3S)-3-(3,4-Dichloro-phenyl)-bi...)
Affinity DataIC50: 22nMAssay Description:In vitro inhibition of [3H]NE re-uptake into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132686(Dimethyl-((2S,3S)-3-naphthalen-2-yl-bicyclo[2.2.1]...)
Affinity DataIC50: 25nMAssay Description:In vitro inhibition of [3H]NE re-uptake into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50026952(CHEMBL322067 | [(2R,3S)-3-(3,4-Dichloro-phenyl)-bi...)
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132679(Methyl-((2S,3S)-3-naphthalen-2-yl-bicyclo[2.2.1]he...)
Affinity DataIC50: 28nMAssay Description:In vitro inhibition of [3H]NE re-uptake into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132677(Dimethyl-((2R,3R)-3-naphthalen-2-yl-bicyclo[2.2.1]...)
Affinity DataIC50: 34nMAssay Description:In vitro inhibition of [3H]NE re-uptake into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132682([(2S,3S)-3-(3-Chloro-phenyl)-bicyclo[2.2.2]oct-2-y...)
Affinity DataIC50: 44nMAssay Description:In vitro inhibition of [3H]NE re-uptake into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132684(Methyl-(3-naphthalen-2-yl-bicyclo[2.2.1]hept-2-ylm...)
Affinity DataIC50: 45nMAssay Description:In vitro inhibition of [3H]NE re-uptake into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132685(Dimethyl-(3-naphthalen-2-yl-bicyclo[2.2.1]hept-2-y...)
Affinity DataIC50: 45nMAssay Description:In vitro inhibition of [3H]NE re-uptake into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132684(Methyl-(3-naphthalen-2-yl-bicyclo[2.2.1]hept-2-ylm...)
Affinity DataIC50: 50nMAssay Description:In vitro ability of compound to inhibit 5-HT re-uptake of radiolabeled [3H]-tritium transmitter into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132686(Dimethyl-((2S,3S)-3-naphthalen-2-yl-bicyclo[2.2.1]...)
Affinity DataIC50: 76nMAssay Description:In vitro inhibition of DA re-uptake into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132679(Methyl-((2S,3S)-3-naphthalen-2-yl-bicyclo[2.2.1]he...)
Affinity DataIC50: 86nMAssay Description:In vitro inhibition of DA re-uptake into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132684(Methyl-(3-naphthalen-2-yl-bicyclo[2.2.1]hept-2-ylm...)
Affinity DataIC50: 87nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132677(Dimethyl-((2R,3R)-3-naphthalen-2-yl-bicyclo[2.2.1]...)
Affinity DataIC50: 93nMAssay Description:In vitro inhibition of DA re-uptake into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132688(Dimethyl-(3-naphthalen-1-yl-bicyclo[2.2.1]hept-2-y...)
Affinity DataIC50: 93nMAssay Description:In vitro ability of compound to inhibit 5-HT re-uptake of radiolabeled [3H]-tritium transmitter into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132685(Dimethyl-(3-naphthalen-2-yl-bicyclo[2.2.1]hept-2-y...)
Affinity DataIC50: 95nMAssay Description:In vitro inhibition of DA re-uptake into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132682([(2S,3S)-3-(3-Chloro-phenyl)-bicyclo[2.2.2]oct-2-y...)
Affinity DataIC50: 165nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50026952(CHEMBL322067 | [(2R,3S)-3-(3,4-Dichloro-phenyl)-bi...)
Affinity DataIC50: 270nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132688(Dimethyl-(3-naphthalen-1-yl-bicyclo[2.2.1]hept-2-y...)
Affinity DataIC50: 297nMAssay Description:In vitro inhibition of [3H]NE re-uptake into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132682([(2S,3S)-3-(3-Chloro-phenyl)-bicyclo[2.2.2]oct-2-y...)
Affinity DataIC50: 303nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132688(Dimethyl-(3-naphthalen-1-yl-bicyclo[2.2.1]hept-2-y...)
Affinity DataIC50: 1.51E+3nMAssay Description:In vitro inhibition of DA re-uptake into synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132686(Dimethyl-((2S,3S)-3-naphthalen-2-yl-bicyclo[2.2.1]...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132687([(2S,3S)-3-(6-Fluoro-naphthalen-2-yl)-bicyclo[2.2....)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132685(Dimethyl-(3-naphthalen-2-yl-bicyclo[2.2.1]hept-2-y...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132679(Methyl-((2S,3S)-3-naphthalen-2-yl-bicyclo[2.2.1]he...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132678([(2S,3S)-3-(6-Fluoro-naphthalen-2-yl)-bicyclo[2.2....)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132684(Methyl-(3-naphthalen-2-yl-bicyclo[2.2.1]hept-2-ylm...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132677(Dimethyl-((2R,3R)-3-naphthalen-2-yl-bicyclo[2.2.1]...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132683(6-((2S,3S)-3-Dimethylaminomethyl-bicyclo[2.2.1]hep...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50026952(CHEMBL322067 | [(2R,3S)-3-(3,4-Dichloro-phenyl)-bi...)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132680([(2S,3S)-3-(6-Methoxy-naphthalen-2-yl)-bicyclo[2.2...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132685(Dimethyl-(3-naphthalen-2-yl-bicyclo[2.2.1]hept-2-y...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132684(Methyl-(3-naphthalen-2-yl-bicyclo[2.2.1]hept-2-ylm...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132681([(2S,3S)-3-(6-Methoxy-naphthalen-2-yl)-bicyclo[2.2...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132682([(2S,3S)-3-(3-Chloro-phenyl)-bicyclo[2.2.2]oct-2-y...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132686(Dimethyl-((2S,3S)-3-naphthalen-2-yl-bicyclo[2.2.1]...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132677(Dimethyl-((2R,3R)-3-naphthalen-2-yl-bicyclo[2.2.1]...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132679(Methyl-((2S,3S)-3-naphthalen-2-yl-bicyclo[2.2.1]he...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50026952(CHEMBL322067 | [(2R,3S)-3-(3,4-Dichloro-phenyl)-bi...)
Affinity DataKi:  44nMAssay Description:Compound was tested for its ability to displace [3H]citalopram from norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132683(6-((2S,3S)-3-Dimethylaminomethyl-bicyclo[2.2.1]hep...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132683(6-((2S,3S)-3-Dimethylaminomethyl-bicyclo[2.2.1]hep...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-Nisoxetine from norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132687([(2S,3S)-3-(6-Fluoro-naphthalen-2-yl)-bicyclo[2.2....)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132682([(2S,3S)-3-(3-Chloro-phenyl)-bicyclo[2.2.2]oct-2-y...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]-Nisoxetine from norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132688(Dimethyl-(3-naphthalen-1-yl-bicyclo[2.2.1]hept-2-y...)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50026952(CHEMBL322067 | [(2R,3S)-3-(3,4-Dichloro-phenyl)-bi...)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132680([(2S,3S)-3-(6-Methoxy-naphthalen-2-yl)-bicyclo[2.2...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132681([(2S,3S)-3-(6-Methoxy-naphthalen-2-yl)-bicyclo[2.2...)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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