Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50036116
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000558(Endothelin-1 | ET-1 | Endothelin -1 | c(Cys-Ser-c(...)
Affinity DataKi:  0.0100nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368606(Sarafotoxin S6B)
Affinity DataKi:  0.0120nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368606(Sarafotoxin S6B)
Affinity DataKi:  0.0130nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000558(Endothelin-1 | ET-1 | Endothelin -1 | c(Cys-Ser-c(...)
Affinity DataKi:  0.0150nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368605(CHEMBL1790178)
Affinity DataKi:  0.0160nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368607(CHEMBL1790180)
Affinity DataKi:  0.0210nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368605(CHEMBL1790178)
Affinity DataKi:  0.0230nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000558(Endothelin-1 | ET-1 | Endothelin -1 | c(Cys-Ser-c(...)
Affinity DataKi:  0.0340nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat atriumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368607(CHEMBL1790180)
Affinity DataKi:  0.0360nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368606(Sarafotoxin S6B)
Affinity DataKi:  0.0870nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat atriumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000558(Endothelin-1 | ET-1 | Endothelin -1 | c(Cys-Ser-c(...)
Affinity DataKi:  0.110nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368606(Sarafotoxin S6B)
Affinity DataKi:  0.240nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat atriumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368607(CHEMBL1790180)
Affinity DataKi:  2.5nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368607(CHEMBL1790180)
Affinity DataKi:  2.5nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000554(CHEMBL432683 | 3-[(2S,5R,8S,11R,14S)-14-(1H-Indol-...)
Affinity DataIC50: 1.40E+3nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the porcine aortic smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000564(CHEMBL538475 | 2-[2-{[2-(Cyclohexanecarbonyl-amino...)
Affinity DataIC50: 2.30E+3nMAssay Description:Compound was evaluated for the binding affinity towards Endothelin A receptor in porcine aortic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000560(CHEMBL37860 | 2-[2-({2-[(Azepane-1-carbonyl)-amino...)
Affinity DataIC50: 2.50E+3nMAssay Description:Compound was evaluated for the binding affinity towards Endothelin A receptor in porcine aortic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000566((S)-3-{(S)-2-[(R)-2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50: 3.70E+3nMAssay Description:Compound was evaluated for the binding affinity to endothelin receptor in the rat heart ventricle.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368605(CHEMBL1790178)
Affinity DataKi:  4.20E+3nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat atriumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368605(CHEMBL1790178)
Affinity DataKi: >5.00E+3nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000559(CHEMBL288514 | 2-(2-Azepan-1-yl-2-oxo-ethyl)-4-met...)
Affinity DataIC50: 7.60E+3nMAssay Description:Compound was evaluated for the binding affinity towards Endothelin A receptor in porcine aortic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000567(CHEMBL287980 | Sodium; ({2-[2-({2-[(azepane-1-carb...)
Affinity DataIC50: 7.60E+3nMAssay Description:Compound was evaluated for the binding affinity towards Endothelin A receptor in porcine aortic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000563(CHEMBL38071 | 3-{2-[2-Acetylamino-3-(3H-imidazol-4...)
Affinity DataIC50: 1.30E+4nMAssay Description:Compound was evaluated for the binding affinity to endothelin receptor in the rat heart ventricle.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000561(CHEMBL290454 | Sodium; 2-{2-[2-({2-[(azepane-1-car...)
Affinity DataIC50: 2.10E+4nMAssay Description:Compound was evaluated for the binding affinity towards Endothelin A receptor in porcine aortic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50329850((R)-3-Amino-4-[(S)-2-((R)-1-{(S)-1-[(R)-1-(1H-indo...)
Affinity DataIC50: 2.20E+4nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the porcine aortic smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Pig)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50329850((R)-3-Amino-4-[(S)-2-((R)-1-{(S)-1-[(R)-1-(1H-indo...)
Affinity DataIC50: 2.30E+4nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the porcine cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000568(CHEMBL431699 | 2-[2-({2-[2-(2-Chloro-phenyl)-acety...)
Affinity DataIC50: 3.20E+4nMAssay Description:Compound was evaluated for the binding affinity towards Endothelin A receptor in porcine aortic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000565((S)-3-{(S)-2-[(S)-2-Amino-3-(3H-imidazol-4-yl)-pro...)
Affinity DataIC50: 4.40E+4nMAssay Description:Compound was evaluated for the binding affinity to endothelin receptor in the rat heart ventricle.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000553((S)-3-{(S)-2-[(S)-2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50: 5.80E+4nMAssay Description:Compound was evaluated for the binding affinity to endothelin receptor in the rat heart ventricle.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Pig)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000554(CHEMBL432683 | 3-[(2S,5R,8S,11R,14S)-14-(1H-Indol-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the porcine cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B/1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000564(CHEMBL538475 | 2-[2-{[2-(Cyclohexanecarbonyl-amino...)
Affinity DataIC50: 2.30E+5nMAssay Description:Compound was evaluated for the Inhibition of the contractile response of Endothelin A receptor in rabbit thoracic aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed