Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50000171
TargetProstacyclin receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50002404(CHEMBL118567 | 9-(3,4,5-Triphenyl-pyrazol-1-yl)-no...)
Affinity DataIC50: 160nMAssay Description:IC50 value was evaluated by measuring the displacement of [3H]iloprost from Prostaglandin I2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50002401(CHEMBL442405 | 8-(4,5-Diphenyl-pyrazol-1-yl)-octan...)
Affinity DataIC50: 160nMAssay Description:IC50 value was evaluated by measuring the displacement of [3H]iloprost from Prostaglandin I2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50002410(9-(3,4-Diphenyl-pyrazol-1-yl)-nonanoic acid | CHEM...)
Affinity DataIC50: 350nMAssay Description:IC50 value was evaluated by measuring the displacement of [3H]iloprost from Prostaglandin I2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50002406(CHEMBL128747 | 9-(4,5-Diphenyl-pyrazol-1-yl)-nonan...)
Affinity DataIC50: 700nMAssay Description:IC50 value was evaluated by measuring the displacement of [3H]iloprost from Prostaglandin I2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50002403(CHEMBL129568 | 9-(3,5-Diphenyl-pyrazol-1-yl)-nonan...)
Affinity DataIC50: 1.00E+4nMAssay Description:IC50 value was evaluated by measuring the displacement of [3H]iloprost from Prostaglandin I2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50002409(CHEMBL129374 | 9-(4-Phenyl-pyrazol-1-yl)-nonanoic ...)
Affinity DataIC50: 1.00E+4nMAssay Description:IC50 value was evaluated by measuring the displacement of [3H]iloprost from Prostaglandin I2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed