Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 5739
TargetProtein kinase C alpha type(Rat)
Mcmaster University

LigandPNGBDBM92971(Amphiphile, VI)
Affinity DataIC50: 1.10E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2013
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Rat)
Mcmaster University

LigandPNGBDBM92969(Amphiphile, IV)
Affinity DataIC50: 1.20E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2013
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Rat)
Mcmaster University

LigandPNGBDBM92976(Amphiphile, XI)
Affinity DataIC50: 1.50E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2013
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Rat)
Mcmaster University

LigandPNGBDBM92978(Amphiphile, XIII)
Affinity DataIC50: 2.00E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2013
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Rat)
Mcmaster University

LigandPNGBDBM92979(Amphiphile, XVI)
Affinity DataIC50: 2.60E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2013
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Rat)
Mcmaster University

LigandPNGBDBM92980(Amphiphile, XVII)
Affinity DataIC50: 4.00E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2013
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Rat)
Mcmaster University

LigandPNGBDBM92974(Amphiphile, IX)
Affinity DataIC50: 5.90E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2013
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Rat)
Mcmaster University

LigandPNGBDBM92977(Amphiphile, XII)
Affinity DataIC50: 1.64E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2013
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Rat)
Mcmaster University

LigandPNGBDBM92973(Amphiphile, VIII)
Affinity DataIC50: 1.91E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2013
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Rat)
Mcmaster University

LigandPNGBDBM92972(Amphiphile, VII)
Affinity DataIC50: 2.46E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2013
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Rat)
Mcmaster University

LigandPNGBDBM92968(Amphiphile, III)
Affinity DataIC50: 2.58E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2013
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Rat)
Mcmaster University

LigandPNGBDBM92975(Amphiphile, X)
Affinity DataIC50: 4.08E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2013
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Rat)
Mcmaster University

LigandPNGBDBM92970(Amphiphile, V)
Affinity DataIC50: 6.43E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2013
Entry Details Article
PubMed