Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50000242
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataIC50: 4nMAssay Description:The compound was tested in vitro for inhibitory activity against 5-HT1A receptor in rats, using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003342(CHEMBL440340 | 6-Bromo-9-methoxy-3-propyl-2,3,4,5-...)
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1A receptor in rats, using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003348(CHEMBL128722 | 6-Methoxy-3-propyl-2,3,4,5-tetrahyd...)
Affinity DataIC50: 63nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1A receptor in rats, using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003346(CHEMBL127221 | 3-Propyl-2,3,4,5-tetrahydro-1H-benz...)
Affinity DataIC50: 81nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1A receptor in rats, using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003345(CHEMBL129293 | 3-Cyclopropylmethyl-6-methoxy-2,3,4...)
Affinity DataIC50: 120nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1A receptor in rats, using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003347(CHEMBL339061 | 3-Ethyl-6-methoxy-2,3,4,5-tetrahydr...)
Affinity DataIC50: 210nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1A receptor in rats, using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003343(CHEMBL132112 | 3-Butyl-2,3,4,5-tetrahydro-1H-benzo...)
Affinity DataIC50: 420nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1A receptor in rats, using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003340(CHEMBL127959 | 6-Methoxy-3-methyl-2,3,4,5-tetrahyd...)
Affinity DataIC50: 480nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1A receptor in rats, using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003341(CHEMBL129249 | 3-Ethyl-2,3,4,5-tetrahydro-1H-benzo...)
Affinity DataIC50: 630nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1A receptor in rats, using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003342(CHEMBL440340 | 6-Bromo-9-methoxy-3-propyl-2,3,4,5-...)
Affinity DataIC50: 680nMAssay Description:The compound was tested in vitro for inhibitory activity against dopamine receptor in rats using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003339(CHEMBL129387 | 3-Methyl-2,3,4,5-tetrahydro-1H-benz...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1A receptor in rats, using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003347(CHEMBL339061 | 3-Ethyl-6-methoxy-2,3,4,5-tetrahydr...)
Affinity DataIC50: 2.20E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against dopamine receptor in rats using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003340(CHEMBL127959 | 6-Methoxy-3-methyl-2,3,4,5-tetrahyd...)
Affinity DataIC50: 2.30E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against dopamine receptor in rats using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003348(CHEMBL128722 | 6-Methoxy-3-propyl-2,3,4,5-tetrahyd...)
Affinity DataIC50: 3.60E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against dopamine receptor in rats using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003344(CHEMBL129676 | 3-Propyl-2,3,4,5-tetrahydro-1H-benz...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1A receptor in rats, using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataIC50: 5.80E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against dopamine receptor in rats using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003345(CHEMBL129293 | 3-Cyclopropylmethyl-6-methoxy-2,3,4...)
Affinity DataIC50: 7.60E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against dopamine receptor in rats using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003344(CHEMBL129676 | 3-Propyl-2,3,4,5-tetrahydro-1H-benz...)
Affinity DataIC50: 1.00E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against dopamine receptor in rats using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003343(CHEMBL132112 | 3-Butyl-2,3,4,5-tetrahydro-1H-benzo...)
Affinity DataIC50: 1.20E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against dopamine receptor in rats using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003341(CHEMBL129249 | 3-Ethyl-2,3,4,5-tetrahydro-1H-benzo...)
Affinity DataIC50: 1.40E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against dopamine receptor in rats using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003339(CHEMBL129387 | 3-Methyl-2,3,4,5-tetrahydro-1H-benz...)
Affinity DataIC50: 1.50E+4nMAssay Description:The compound was tested in vitro for inhibitory activity against dopamine receptor in rats using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50003346(CHEMBL127221 | 3-Propyl-2,3,4,5-tetrahydro-1H-benz...)
Affinity DataIC50: 1.00E+5nMAssay Description:The compound was tested in vitro for inhibitory activity against dopamine receptor in rats using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed