Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50000260
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003669(CHEMBL411079 | Ac-Tyr(SO3H)-Met-Gly-Trp-Met-R-Dtc-...)
Affinity DataIC50: 0.0500nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003666(3-[2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 0.0500nMAssay Description:Inhibitory activity against cholecystokinin type A receptor from rat pancreas binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003670(3-{2-[2-(2-{2-[2-Acetylamino-3-(4-sulfo-phenyl)-pr...)
Affinity DataIC50: 0.600nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003667(4-{2-Acetylamino-2-[1-({[1-{1-[2-carbamoyl-1-(1-ca...)
Affinity DataIC50: 1.40nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003664(4-{2-Acetylamino-2-[1-({[1-{1-[1-(1-carbamoyl-2-ph...)
Affinity DataIC50: 2.40nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Bovine)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003670(3-{2-[2-(2-{2-[2-Acetylamino-3-(4-sulfo-phenyl)-pr...)
Affinity DataIC50: 4.40nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003665(3-{2-[2-(2-{2-[2-Acetylamino-3-(4-sulfo-phenyl)-pr...)
Affinity DataIC50: 5.5nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003662(4-{2-Acetylamino-2-[1-({[1-{1-[2-(1-carbamoyl-2-ph...)
Affinity DataIC50: 8.30nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Bovine)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003665(3-{2-[2-(2-{2-[2-Acetylamino-3-(4-sulfo-phenyl)-pr...)
Affinity DataIC50: 22nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003668([1-[1-[4-(1-Carbamoyl-2-phenyl-ethylcarbamoyl)-5,5...)
Affinity DataIC50: 59nMAssay Description:Inhibitory activity against cholecystokinin type A receptor from rat pancreas binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Bovine)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003664(4-{2-Acetylamino-2-[1-({[1-{1-[1-(1-carbamoyl-2-ph...)
Affinity DataIC50: 170nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Bovine)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003667(4-{2-Acetylamino-2-[1-({[1-{1-[2-carbamoyl-1-(1-ca...)
Affinity DataIC50: 200nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003663(CHEMBL385727 | Ac-Tyr(SO3H)-Met-Gly-Trp-Met-S-Dtc-...)
Affinity DataIC50: 314nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003666(3-[2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity against cholecystokinin type A receptor from bovine striatal binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Bovine)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003669(CHEMBL411079 | Ac-Tyr(SO3H)-Met-Gly-Trp-Met-R-Dtc-...)
Affinity DataIC50: 2.31E+3nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Bovine)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003662(4-{2-Acetylamino-2-[1-({[1-{1-[2-(1-carbamoyl-2-ph...)
Affinity DataIC50: 3.90E+3nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Bovine)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003663(CHEMBL385727 | Ac-Tyr(SO3H)-Met-Gly-Trp-Met-S-Dtc-...)
Affinity DataIC50: 6.16E+3nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003668([1-[1-[4-(1-Carbamoyl-2-phenyl-ethylcarbamoyl)-5,5...)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibitory activity against cholecystokinin type A receptor from bovine striatal binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed