Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50013782
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50204884(6-(2-(4-(4-fluorobenzyl)piperidin-1-yl)ethylsulfin...)
Affinity DataIC50: 8nMAssay Description:Inhibition of N-methyl-D-aspartate glutamate receptor-evoked increase of intracellular Ca+ in cells expressing NMDA glutamate receptor 1/2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50134652((4-benzylpiperidine-1-yl)-(4,6-dihydroxy-1H-indole...)
Affinity DataIC50: 10nMAssay Description:Inhibition of N-methyl-D-aspartate glutamate receptor-evoked increase of intracellular Ca+ in cells expressing NMDA glutamate receptor 1/2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50134648((6-hydroxy-1H-indole-2-yl)-(4-phenoxymethylpiperid...)
Affinity DataIC50: 19nMAssay Description:Inhibition of N-methyl-D-aspartate glutamate receptor-evoked increase of intracellular Ca+ in cells expressing NMDA glutamate receptor 1/2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50134651((4-Benzyl-piperidin-1-yl)-(6-hydroxy-1H-indol-2-yl...)
Affinity DataIC50: 20nMAssay Description:Inhibition of N-methyl-D-aspartate glutamate receptor-evoked increase of intracellular Ca+ in cells expressing NMDA glutamate receptor 1/2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50134649((6-hydroxy-1H-indole-2-yl)-(4-phenylethylpiperidin...)
Affinity DataIC50: 24nMAssay Description:Inhibition of N-methyl-D-aspartate glutamate receptor-evoked increase of intracellular Ca+ in cells expressing NMDA glutamate receptor 1/2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50134653((4-Benzyl-piperidin-1-yl)-(4-hydroxy-1H-indol-2-yl...)
Affinity DataIC50: 39nMAssay Description:Inhibition of N-methyl-D-aspartate glutamate receptor-evoked increase of intracellular Ca+ in cells expressing NMDA glutamate receptor 1/2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50134657((4-Benzyl-piperidin-1-yl)-(5-hydroxy-1H-indol-2-yl...)
Affinity DataIC50: 40nMAssay Description:Inhibition of N-methyl-D-aspartate glutamate receptor-evoked increase of intracellular Ca+ in cells expressing NMDA glutamate receptor 1/2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50134656((4-Benzyloxy-piperidin-1-yl)-(6-hydroxy-1H-indol-2...)
Affinity DataIC50: 46nMAssay Description:Inhibition of N-methyl-D-aspartate glutamate receptor-evoked increase of intracellular Ca+ in cells expressing NMDA glutamate receptor 1/2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50134654((4-Benzyl-piperidin-1-yl)-(5,7-dihydroxy-1H-indol-...)
Affinity DataIC50: 52nMAssay Description:Inhibition of N-methyl-D-aspartate glutamate receptor-evoked increase of intracellular Ca+ in cells expressing NMDA glutamate receptor 1/2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50080029(CHEMBL305195 | 4-[(1R,2S)-3-(4-Benzyl-piperidin-1-...)
Affinity DataIC50: 57nMAssay Description:Inhibition of N-methyl-D-aspartate glutamate receptor-evoked increase of intracellular Ca+ in cells expressing NMDA glutamate receptor 1/2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50134650((4-benzylpiperidin-1-yl)(7-hydroxy-1H-indol-2-yl)m...)
Affinity DataIC50: 77nMAssay Description:Inhibition of N-methyl-D-aspartate glutamate receptor-evoked increase of intracellular Ca+ in cells expressing NMDA glutamate receptor 1/2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50080016((E)-1-(4-Benzyl-piperidin-1-yl)-3-(4-hydroxy-pheny...)
Affinity DataIC50: 104nMAssay Description:Inhibition of N-methyl-D-aspartate glutamate receptor-evoked increase of intracellular Ca+ in cells expressing NMDA glutamate receptor 1/2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50134655((6-hydroxy-1H-indole-2-yl)-(4-phenylpiperidine-1-y...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of N-methyl-D-aspartate glutamate receptor-evoked increase of intracellular Ca+ in cells expressing NMDA glutamate receptor 1/2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed