Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50013915
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Morphochem

Curated by ChEMBL
LigandPNGBDBM21690(Ciprinol | 1-cyclopropyl-6-fluoro-4-oxo-7-(piperaz...)
Affinity DataIC50: 500nMAssay Description:Inhibitory activity against DNA gyrase enzyme was determined by supercoiling assay with Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Morphochem

Curated by ChEMBL
LigandPNGBDBM50135931(7-(3-{4-[(S)-5-(Acetylamino-methyl)-2-oxo-oxazolid...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against DNA gyrase enzyme was determined by supercoiling assay with Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Morphochem

Curated by ChEMBL
LigandPNGBDBM50135930(7-((S)-3-{4-[(S)-5-(Acetylamino-methyl)-2-oxo-oxaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against DNA gyrase enzyme was determined by supercoiling assay with Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Morphochem

Curated by ChEMBL
LigandPNGBDBM50135928(7-(4-{4-[(S)-5-(Acetylamino-methyl)-2-oxo-oxazolid...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against DNA gyrase enzyme was determined by supercoiling assay with Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Morphochem

Curated by ChEMBL
LigandPNGBDBM50135929(7-(4-{4-[(S)-5-(Acetylamino-methyl)-2-oxo-oxazolid...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against DNA gyrase enzyme was determined by supercoiling assay with Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed