Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 2158
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17589(bestatin-type inhibitor, 4 | CHEMBL352943 | (2S,3R...)
Affinity DataIC50: 22nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17590(CHEMBL171479 | (2S,3S)-3-amino-2-hydroxy-4-[(2-met...)
Affinity DataIC50: 48nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17592(N'-[(2S,3R)-3-amino-5-(ethylsulfanyl)-2-hydroxypen...)
Affinity DataIC50: 110nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17594(N'-[(2S,3R)-3-amino-2-hydroxy-5-(propan-2-ylsulfan...)
Affinity DataIC50: 120nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17593(CHEMBL170733 | N'-[(2S,3S)-3-amino-2-hydroxy-4-[(2...)
Affinity DataIC50: 130nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17591(CHEMBL170271 | (2S,3R)-3-amino-2-hydroxy-N-[(1S)-1...)
Affinity DataIC50: 190nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 1(Human)
Abbott Laboratories

LigandPNGBDBM17589(bestatin-type inhibitor, 4 | CHEMBL352943 | (2S,3R...)
Affinity DataIC50: 370nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17588(ethyl (2S)-2-[(2S,3S)-3-amino-2-hydroxy-4-[(2-meth...)
Affinity DataIC50: 1.10E+3nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17587(ethyl (2S)-2-[(2S,3R)-3-amino-5-(ethylsulfanyl)-2-...)
Affinity DataIC50: 1.30E+3nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 1(Human)
Abbott Laboratories

LigandPNGBDBM17590(CHEMBL171479 | (2S,3S)-3-amino-2-hydroxy-4-[(2-met...)
Affinity DataIC50: 2.20E+3nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17586(ethyl (2S)-2-[(2S,3R)-3-amino-2-hydroxy-5-(methyls...)
Affinity DataIC50: 6.00E+3nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 1(Human)
Abbott Laboratories

LigandPNGBDBM17593(CHEMBL170733 | N'-[(2S,3S)-3-amino-2-hydroxy-4-[(2...)
Affinity DataIC50: 8.10E+3nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 1(Human)
Abbott Laboratories

LigandPNGBDBM17591(CHEMBL170271 | (2S,3R)-3-amino-2-hydroxy-N-[(1S)-1...)
Affinity DataIC50: 1.20E+4nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 1(Human)
Abbott Laboratories

LigandPNGBDBM17592(N'-[(2S,3R)-3-amino-5-(ethylsulfanyl)-2-hydroxypen...)
Affinity DataIC50: 2.00E+4nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 1(Human)
Abbott Laboratories

LigandPNGBDBM17594(N'-[(2S,3R)-3-amino-2-hydroxy-5-(propan-2-ylsulfan...)
Affinity DataIC50: 5.70E+4nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 1(Human)
Abbott Laboratories

LigandPNGBDBM17586(ethyl (2S)-2-[(2S,3R)-3-amino-2-hydroxy-5-(methyls...)
Affinity DataIC50: 6.30E+4nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 1(Human)
Abbott Laboratories

LigandPNGBDBM17588(ethyl (2S)-2-[(2S,3S)-3-amino-2-hydroxy-4-[(2-meth...)
Affinity DataIC50: 6.60E+4nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 1(Human)
Abbott Laboratories

LigandPNGBDBM17587(ethyl (2S)-2-[(2S,3R)-3-amino-5-(ethylsulfanyl)-2-...)
Affinity DataIC50: 6.90E+4nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed