Compile Data Set for Download or QSAR
Report error Found 71 Enz. Inhib. hit(s) with all data for entry = 50013967
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136445(5-Chloro-1H-indole-2-carboxylic acid ((R)-2-oxo-1,...)
Affinity DataIC50: 14nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136451(5-Chloro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50: 25nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136445(5-Chloro-1H-indole-2-carboxylic acid ((R)-2-oxo-1,...)
Affinity DataIC50: 25nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136440(5-Bromo-1H-indole-2-carboxylic acid (1-methyl-2-ox...)
Affinity DataIC50: 30nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136451(5-Chloro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50: 32nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136437(5-chloro-N-(2-oxo-1,2,3,4-tetrahydroquinolin-3-yl)...)
Affinity DataIC50: 38nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136447(5-Chloro-1H-indole-2-carboxylic acid ((S)-2-oxo-1,...)
Affinity DataIC50: 39nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136437(5-chloro-N-(2-oxo-1,2,3,4-tetrahydroquinolin-3-yl)...)
Affinity DataIC50: 44nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136446([5-CHLORO-1H-INDOL-2-CARBONYL-PHENYLALANINYL]-AZET...)
Affinity DataIC50: 45nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136447(5-Chloro-1H-indole-2-carboxylic acid ((S)-2-oxo-1,...)
Affinity DataIC50: 47nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136424(5-Chloro-7-fluoro-1H-indole-2-carboxylic acid (1-m...)
Affinity DataIC50: 55nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136435(5-Chloro-1H-indole-2-carboxylic acid (2-oxo-2,3,4,...)
Affinity DataIC50: 55nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136418(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-1,2,3,...)
Affinity DataIC50: 56nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136428(5-Chloro-1H-indole-2-carboxylic acid ((S)-1-methyl...)
Affinity DataIC50: 57nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136428(5-Chloro-1H-indole-2-carboxylic acid ((S)-1-methyl...)
Affinity DataIC50: 57nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136448(5-Chloro-1H-indole-2-carboxylic acid ((R)-1-methyl...)
Affinity DataIC50: 58nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136448(5-Chloro-1H-indole-2-carboxylic acid ((R)-1-methyl...)
Affinity DataIC50: 61nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136416(6-Chloro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50: 69nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136440(5-Bromo-1H-indole-2-carboxylic acid (1-methyl-2-ox...)
Affinity DataIC50: 73nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136424(5-Chloro-7-fluoro-1H-indole-2-carboxylic acid (1-m...)
Affinity DataIC50: 83nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136430(5-Chloro-1H-indole-2-carboxylic acid ((R)-2-oxo-2,...)
Affinity DataIC50: 83nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136450(7-Chloro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50: 88nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136450(7-Chloro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50: 88nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136414(5-Fluoro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50: 89nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136443(5-Methyl-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50: 98nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136430(5-Chloro-1H-indole-2-carboxylic acid ((R)-2-oxo-2,...)
Affinity DataIC50: 99nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136416(6-Chloro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50: 99nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136435(5-Chloro-1H-indole-2-carboxylic acid (2-oxo-2,3,4,...)
Affinity DataIC50: 105nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136444(5-Chloro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50: 105nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136417(5-Cyano-1H-indole-2-carboxylic acid (1-methyl-2-ox...)
Affinity DataIC50: 110nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136425(5-Chloro-1H-indole-2-carboxylic acid (2-oxo-1-pyri...)
Affinity DataIC50: 110nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136443(5-Methyl-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50: 120nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136434(7-Nitro-1H-indole-2-carboxylic acid (1-methyl-2-ox...)
Affinity DataIC50: 120nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136414(5-Fluoro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50: 120nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136423(5-Chloro-1H-indole-2-carboxylic acid ((R)-2-oxo-1-...)
Affinity DataIC50: 120nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136420(5-Chloro-1H-indole-2-carboxylic acid (2-oxo-1-pyri...)
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136429(5-Chloro-1H-indole-2-carboxylic acid [1-(5-methyl-...)
Affinity DataIC50: 140nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136436(5-Chloro-1H-indole-2-carboxylic acid ((S)-2-oxo-1-...)
Affinity DataIC50: 140nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136418(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-1,2,3,...)
Affinity DataIC50: 160nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136441(5-Chloro-1H-indole-2-carboxylic acid {1-[5-(1H-imi...)
Affinity DataIC50: 160nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136417(5-Cyano-1H-indole-2-carboxylic acid (1-methyl-2-ox...)
Affinity DataIC50: 180nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136442(5-Chloro-1H-indole-2-carboxylic acid ((S)-2-oxo-2,...)
Affinity DataIC50: 240nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136442(5-Chloro-1H-indole-2-carboxylic acid ((S)-2-oxo-2,...)
Affinity DataIC50: 240nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136434(7-Nitro-1H-indole-2-carboxylic acid (1-methyl-2-ox...)
Affinity DataIC50: 300nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136444(5-Chloro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50: 305nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136449(5-Trifluoromethyl-1H-indole-2-carboxylic acid (1-m...)
Affinity DataIC50: 550nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136438(5-Ethyl-1H-indole-2-carboxylic acid (1-methyl-2-ox...)
Affinity DataIC50: 850nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136421(1H-Indole-2-carboxylic acid (2-oxo-2,3,4,5-tetrahy...)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136433(7-Amino-1H-indole-2-carboxylic acid (1-methyl-2-ox...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136419(3,4-Dichloro-N-(2-oxo-1,2,3,4-tetrahydro-quinolin-...)
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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