Compile Data Set for Download or QSAR
Report error Found 107 Enz. Inhib. hit(s) with all data for entry = 50034691
Target5-hydroxytryptamine receptor 2A(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50007568(CHEMBL303313 | 1-(8-Chloro-10,11-dihydro-dibenzo[b...)
Affinity DataKi:  0.140nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2A receptor in rat tissue homogenate using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137975(7-Bromo-9-(4-methyl-piperazin-1-yl)-4-thia-10a-aza...)
Affinity DataKi:  0.25nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 in Sf9 cell membranes using [3H]7-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50007567(CHEMBL64875 | OCTOCLOTHEPIN-R | 1-(8-Chloro-10,11-...)
Affinity DataKi:  0.330nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2A receptor in rat tissue homogenate using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137981(7-Chloro-9-(4-methyl-piperazin-1-yl)-4-thia-10a-az...)
Affinity DataKi:  0.340nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2A receptor in rat tissue homogenate using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137972(7-Fluoro-9-(4-methyl-piperazin-1-yl)-4-thia-10a-az...)
Affinity DataKi:  0.350nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2A receptor in rat tissue homogenate using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50007568(CHEMBL303313 | 1-(8-Chloro-10,11-dihydro-dibenzo[b...)
Affinity DataKi:  0.400nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 in Sf9 cell membranes using [3H]7-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50007568(CHEMBL303313 | 1-(8-Chloro-10,11-dihydro-dibenzo[b...)
Affinity DataKi:  0.400nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 in rat tissue homogenate using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137981(7-Chloro-9-(4-methyl-piperazin-1-yl)-4-thia-10a-az...)
Affinity DataKi:  0.430nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 in rat tissue homogenate using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137975(7-Bromo-9-(4-methyl-piperazin-1-yl)-4-thia-10a-aza...)
Affinity DataKi:  0.450nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 in rat tissue homogenate using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137976(9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f...)
Affinity DataKi:  0.5nMAssay Description:In vitro binding affinity towards alpha-1 adrenergic receptor in rat frontal cortex homogenate using of [3H]prazosin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137976(9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f...)
Affinity DataKi:  0.650nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2A receptor in rat tissue homogenate using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137978((S)-7-Chloro-9-(4-methyl-piperazin-1-yl)-9,10-dihy...)
Affinity DataKi:  0.820nMAssay Description:In vitro binding affinity towards alpha-1 adrenergic receptor in rat frontal cortex homogenate using of [3H]prazosin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137975(7-Bromo-9-(4-methyl-piperazin-1-yl)-4-thia-10a-aza...)
Affinity DataKi:  0.830nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2A receptor in rat tissue homogenate using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50028601(1-(8-Chloro-5H-dibenzo[a,d]cyclohepten-10-yl)-4-me...)
Affinity DataKi:  1nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 in rat tissue homogenate using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137976(9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f...)
Affinity DataKi:  1.10nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2A receptor in human using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137980(1-Methyl-9-(4-methyl-piperazin-1-yl)-4-thia-10a-az...)
Affinity DataKi:  1.10nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2A receptor in rat tissue homogenate using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137978((S)-7-Chloro-9-(4-methyl-piperazin-1-yl)-9,10-dihy...)
Affinity DataKi:  1.5nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2A receptor in rat tissue homogenate using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50007568(CHEMBL303313 | 1-(8-Chloro-10,11-dihydro-dibenzo[b...)
Affinity DataKi:  1.90nMAssay Description:In vitro binding affinity towards Dopamine receptor D1 in rat tissue homogenate using [3H]-SCH- 23390 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137981(7-Chloro-9-(4-methyl-piperazin-1-yl)-4-thia-10a-az...)
Affinity DataKi:  1.90nMAssay Description:In vitro binding affinity towards Dopamine receptor D1 in rat tissue homogenate using [3H]-SCH- 23390 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137981(7-Chloro-9-(4-methyl-piperazin-1-yl)-4-thia-10a-az...)
Affinity DataKi:  2nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 in Sf9 cell membranes using [3H]7-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50007567(CHEMBL64875 | OCTOCLOTHEPIN-R | 1-(8-Chloro-10,11-...)
Affinity DataKi:  2nMAssay Description:In vitro binding affinity towards Dopamine receptor D1 in rat tissue homogenate using [3H]-SCH- 23390 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137972(7-Fluoro-9-(4-methyl-piperazin-1-yl)-4-thia-10a-az...)
Affinity DataKi:  2.70nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 in Sf9 cell membranes using [3H]7-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137980(1-Methyl-9-(4-methyl-piperazin-1-yl)-4-thia-10a-az...)
Affinity DataKi:  2.70nMAssay Description:In vitro binding affinity towards Histamine H1 receptor of rat frontal cortex homogenate by using radioligand [3H]pyrilamineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137976(9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f...)
Affinity DataKi:  2.70nMAssay Description:In vitro binding affinity towards Histamine H1 receptor of rat frontal cortex homogenate by using radioligand [3H]pyrilamineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  2.90nMAssay Description:In vitro binding affinity towards Histamine H1 receptor of rat frontal cortex homogenate by using radioligand [3H]pyrilamineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137975(7-Bromo-9-(4-methyl-piperazin-1-yl)-4-thia-10a-aza...)
Affinity DataKi:  3.40nMAssay Description:In vitro binding affinity towards Dopamine receptor D1 in rat tissue homogenate using [3H]-SCH- 23390 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137982(7-Chloro-9-(4-methyl-[1,4]diazepan-1-yl)-4-thia-10...)
Affinity DataKi:  3.5nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 in rat tissue homogenate using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50007567(CHEMBL64875 | OCTOCLOTHEPIN-R | 1-(8-Chloro-10,11-...)
Affinity DataKi:  3.60nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 in rat tissue homogenate using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  3.70nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 in human using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM35254(CHEMBL715 | 2-methyl-4-(4-methylpiperazin-1-yl)-10...)
Affinity DataKi:  4nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2A receptor in rat tissue homogenate using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137980(1-Methyl-9-(4-methyl-piperazin-1-yl)-4-thia-10a-az...)
Affinity DataKi:  4.20nMAssay Description:In vitro binding affinity towards alpha-1 adrenergic receptor in rat frontal cortex homogenate using of [3H]prazosin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137982(7-Chloro-9-(4-methyl-[1,4]diazepan-1-yl)-4-thia-10...)
Affinity DataKi:  4.30nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2A receptor in rat tissue homogenate using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM35254(CHEMBL715 | 2-methyl-4-(4-methylpiperazin-1-yl)-10...)
Affinity DataKi:  4.30nMAssay Description:In vitro binding affinity towards Histamine H1 receptor of rat frontal cortex homogenate by using radioligand [3H]pyrilamineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137982(7-Chloro-9-(4-methyl-[1,4]diazepan-1-yl)-4-thia-10...)
Affinity DataKi:  4.30nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 in Sf9 cell membranes using [3H]7-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  4.80nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 in rat tissue homogenate using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137982(7-Chloro-9-(4-methyl-[1,4]diazepan-1-yl)-4-thia-10...)
Affinity DataKi:  5.90nMAssay Description:In vitro binding affinity towards Dopamine receptor D1 in rat tissue homogenate using [3H]-SCH- 23390 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137972(7-Fluoro-9-(4-methyl-piperazin-1-yl)-4-thia-10a-az...)
Affinity DataKi:  7.70nMAssay Description:In vitro binding affinity towards Dopamine receptor D1 in rat tissue homogenate using [3H]-SCH- 23390 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  7.80nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2A receptor in human using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137976(9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f...)
Affinity DataKi:  8.30nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 in Sf9 cell membranes using [3H]7-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137972(7-Fluoro-9-(4-methyl-piperazin-1-yl)-4-thia-10a-az...)
Affinity DataKi:  8.5nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 in rat tissue homogenate using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  9nMAssay Description:In vitro binding affinity towards alpha-1 adrenergic receptor in rat frontal cortex homogenate using of [3H]prazosin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  10nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2A receptor in rat tissue homogenate using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  12nMAssay Description:In vitro binding affinity towards alpha-1 adrenergic receptor in rat frontal cortex homogenate using of [3H]prazosin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137976(9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f...)
Affinity DataKi:  13nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 in human using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM35254(CHEMBL715 | 2-methyl-4-(4-methylpiperazin-1-yl)-10...)
Affinity DataKi:  15nMAssay Description:In vitro binding affinity towards alpha-1 adrenergic receptor in rat frontal cortex homogenate using of [3H]prazosin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137978((S)-7-Chloro-9-(4-methyl-piperazin-1-yl)-9,10-dihy...)
Affinity DataKi:  16nMAssay Description:In vitro binding affinity towards Dopamine receptor D1 in rat tissue homogenate using [3H]-SCH- 23390 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137976(9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f...)
Affinity DataKi:  17nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 in rat tissue homogenate using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137976(9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f...)
Affinity DataKi:  17nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 in rat tissue homogenate using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50137980(1-Methyl-9-(4-methyl-piperazin-1-yl)-4-thia-10a-az...)
Affinity DataKi:  18nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 in Sf9 cell membranes using [3H]7-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  18nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 in Sf9 cell membranes using [3H]7-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article
PubMed
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