Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50014110
LigandPNGBDBM50138394(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-...)
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138386(1-[5-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyri...)
Affinity DataIC50: 26nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138381((4-Methanesulfonyl-phenyl)-{4-[4-(piperazine-1-sul...)
Affinity DataIC50: 31nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138384(N-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimid...)
Affinity DataIC50: 43nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138400(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-...)
Affinity DataIC50: 44nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138391(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-...)
Affinity DataIC50: 48nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138380(1-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimid...)
Affinity DataIC50: 59nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138398((4-Benzothiazol-6-yl-phenyl)-{4-[4-(piperazine-1-s...)
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138393((4-Nitro-phenyl)-{4-[4-(piperazine-1-sulfonyl)-phe...)
Affinity DataIC50: 66nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138396(3-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-...)
Affinity DataIC50: 83nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138395(Phenyl-{4-[4-(piperazine-1-sulfonyl)-phenyl]-pyrim...)
Affinity DataIC50: 91nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138385((4-Methanesulfinyl-phenyl)-{4-[4-(piperazine-1-sul...)
Affinity DataIC50: 91nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138392((3,4-Difluoro-phenyl)-{4-[4-(piperazine-1-sulfonyl...)
Affinity DataIC50: 117nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138383({4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-...)
Affinity DataIC50: 145nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138390((4-Chloro-phenyl)-{4-[4-(piperazine-1-sulfonyl)-ph...)
Affinity DataIC50: 148nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138383({4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-...)
Affinity DataIC50: 155nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138397((4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin...)
Affinity DataIC50: 155nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138399((4-Methoxy-phenyl)-{4-[4-(piperazine-1-sulfonyl)-p...)
Affinity DataIC50: 214nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138394(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-...)
Affinity DataIC50: 245nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138401({4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-...)
Affinity DataIC50: 269nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138388((4-Butyl-phenyl)-{4-[4-(piperazine-1-sulfonyl)-phe...)
Affinity DataIC50: 309nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138384(N-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimid...)
Affinity DataIC50: 331nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138387(N-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimid...)
Affinity DataIC50: 331nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138389({4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-...)
Affinity DataIC50: 513nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138382(5-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimid...)
Affinity DataIC50: 550nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138382(5-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimid...)
Affinity DataIC50: 550nMAssay Description:Inhibitory activity against IKK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138398((4-Benzothiazol-6-yl-phenyl)-{4-[4-(piperazine-1-s...)
Affinity DataIC50: 851nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138380(1-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimid...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138395(Phenyl-{4-[4-(piperazine-1-sulfonyl)-phenyl]-pyrim...)
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138381((4-Methanesulfonyl-phenyl)-{4-[4-(piperazine-1-sul...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138399((4-Methoxy-phenyl)-{4-[4-(piperazine-1-sulfonyl)-p...)
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138397((4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin...)
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138387(N-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimid...)
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138386(1-[5-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyri...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138401({4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-...)
Affinity DataIC50: 2.09E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138385((4-Methanesulfinyl-phenyl)-{4-[4-(piperazine-1-sul...)
Affinity DataIC50: 2.34E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138390((4-Chloro-phenyl)-{4-[4-(piperazine-1-sulfonyl)-ph...)
Affinity DataIC50: 2.34E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138388((4-Butyl-phenyl)-{4-[4-(piperazine-1-sulfonyl)-phe...)
Affinity DataIC50: 2.69E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138382(5-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimid...)
Affinity DataIC50: 3.09E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138382(5-(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimid...)
Affinity DataIC50: 3.09E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138400(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138389({4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-2-...)
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138391(4-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-...)
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138392((3,4-Difluoro-phenyl)-{4-[4-(piperazine-1-sulfonyl...)
Affinity DataIC50: 4.07E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138396(3-{4-[4-(Piperazine-1-sulfonyl)-phenyl]-pyrimidin-...)
Affinity DataIC50: 5.13E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50138393((4-Nitro-phenyl)-{4-[4-(piperazine-1-sulfonyl)-phe...)
Affinity DataIC50: 6.92E+3nMAssay Description:Inhibitory activity against IKK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed