Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 1505
LigandPNGBDBM11823(N-[(3R,4R)-4-({4-[(2-fluoro-6-hydroxy-3-methoxyphe...)
Affinity DataIC50: 2nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2006
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Roche Diagnostics

LigandPNGBDBM11823(N-[(3R,4R)-4-({4-[(2-fluoro-6-hydroxy-3-methoxyphe...)
Affinity DataIC50: 4nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2006
Entry Details Article
PubMed
LigandPNGBDBM11822((3R,4R)-3-(pyridine-4-amido)azepan-4-yl 4-[(2-fluo...)
Affinity DataIC50: 5nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2006
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Roche Diagnostics

LigandPNGBDBM11822((3R,4R)-3-(pyridine-4-amido)azepan-4-yl 4-[(2-fluo...)
Affinity DataIC50: 5nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2006
Entry Details Article
PubMed
LigandPNGBDBM11824(N-((3R,4R)-4-{[4-(2-fluoro-6-hydroxy-3-methoxybenz...)
Affinity DataIC50: 39nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2006
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Roche Diagnostics

LigandPNGBDBM11827(N-[(3S,4S)-4-[(E)-2-{4-[(2-fluoro-6-hydroxy-3-meth...)
Affinity DataIC50: 160nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2006
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Roche Diagnostics

LigandPNGBDBM11824(N-((3R,4R)-4-{[4-(2-fluoro-6-hydroxy-3-methoxybenz...)
Affinity DataIC50: 355nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2006
Entry Details Article
PubMed
LigandPNGBDBM11827(N-[(3S,4S)-4-[(E)-2-{4-[(2-fluoro-6-hydroxy-3-meth...)
Affinity DataIC50: 360nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2006
Entry Details Article
PubMed
LigandPNGBDBM11826(N-((3R,4R)-4-{[4-(2-fluoro-6-hydroxy-3-methoxybenz...)
Affinity DataIC50: 800nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2006
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Roche Diagnostics

LigandPNGBDBM11826(N-((3R,4R)-4-{[4-(2-fluoro-6-hydroxy-3-methoxybenz...)
Affinity DataIC50: 3.00E+3nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2006
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Roche Diagnostics

LigandPNGBDBM11825(N-[(3S,4S)-4-[({4-[(2-fluoro-6-hydroxy-3-methoxyph...)
Affinity DataIC50: 2.50E+4nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2006
Entry Details Article
PubMed
LigandPNGBDBM11825(N-[(3S,4S)-4-[({4-[(2-fluoro-6-hydroxy-3-methoxyph...)
Affinity DataIC50: 4.50E+4nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2006
Entry Details Article
PubMed