Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50014444
LigandPNGBDBM50090540(7-Chloro-2-oxo-4-((S)-2-piperidin-2-yl-ethoxy)-3-(...)
Affinity DataIC50: 0.300nMAssay Description:Inhibitory concentration against binding of [125I]buserelin to human Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50142827(7-Chloro-3-(3,5-dimethyl-phenyl)-4-[2-((S)-(S)-6-m...)
Affinity DataIC50: 0.5nMAssay Description:Inhibitory concentration against binding of [125I]buserelin to human Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50142834(7-Chloro-3-(3,5-dimethyl-phenyl)-4-[2-((S)-(R)-6-m...)
Affinity DataIC50: 0.5nMAssay Description:Inhibitory concentration against binding of [125I]buserelin to human Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50142826(7-Chloro-3-((S)-3,5-dimethyl-4-methyl-phenyl)-4-[2...)
Affinity DataIC50: 0.600nMAssay Description:Inhibitory concentration against binding of [125I]buserelin to human Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50142829(7-Chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-((S)-2-pi...)
Affinity DataIC50: 0.900nMAssay Description:Inhibitory concentration against binding of [125I]buserelin to human Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50142828(7-Chloro-2-oxo-4-[2-((S)-6-trifluoromethyl-piperid...)
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against binding of [125I]buserelin to human Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50142832(7-Chloro-3-(3,5-dimethyl-phenyl)-4-[2-((S)-6-ethyl...)
Affinity DataIC50: 5.70nMAssay Description:Inhibitory concentration against binding of [125I]buserelin to human Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50081148(CHEMBL294910 | CHEMBL90725 | 7-Chloro-3-(3,5-dimet...)
Affinity DataIC50: 10nMAssay Description:Inhibitory concentration against binding of rat Gonadotropin-releasing hormone receptor using [125I]buserelinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50081148(CHEMBL294910 | CHEMBL90725 | 7-Chloro-3-(3,5-dimet...)
Affinity DataIC50: 10nMAssay Description:Inhibitory concentration against binding of rat Gonadotropin-releasing hormone receptor using [125I]buserelinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50404356(CHEMBL2113717)
Affinity DataIC50: 15nMAssay Description:Inhibitory concentration against binding of rat Gonadotropin-releasing hormone receptor using [125I]buserelinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50404355(CHEMBL2113716)
Affinity DataIC50: 18nMAssay Description:Inhibitory concentration against binding of rat Gonadotropin-releasing hormone receptor using [125I]buserelinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50142837(7-Chloro-3-(3,5-dimethyl-phenyl)-4-[2-(3-methyl-pi...)
Affinity DataIC50: 45nMAssay Description:Inhibitory concentration against binding of rat Gonadotropin-releasing hormone receptor using [125I]buserelinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50142833(7-Chloro-3-(3,5-dimethyl-phenyl)-4-[2-(5-methyl-pi...)
Affinity DataIC50: 63nMAssay Description:Inhibitory concentration against binding of rat Gonadotropin-releasing hormone receptor using [125I]buserelinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50142835(7-Chloro-3-(3,5-dimethyl-phenyl)-6-nitro-4-[(S)-2-...)
Affinity DataIC50: 70nMAssay Description:Inhibitory concentration against binding of rat Gonadotropin-releasing hormone receptor using [125I]buserelinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50404354(CHEMBL2113713)
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration against binding of rat Gonadotropin-releasing hormone receptor using [125I]buserelinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50142831(7-Chloro-3-(3,5-dimethyl-phenyl)-6-nitro-4-[2-(1,2...)
Affinity DataIC50: 750nMAssay Description:Inhibitory concentration against binding of rat Gonadotropin-releasing hormone receptor using [125I]buserelinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed