Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50014445
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Potency of inhibiting 10 pM [125I]-RTI-55 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Potency of inhibiting [3H]WIN-35428 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Potency of inhibiting [3H]WIN-35428 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Potency of inhibiting [3H]WIN-35428 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 33.9nMAssay Description:Potency of inhibiting 10 pM [125I]-RTI-55 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Potency of inhibiting 10 pM [125I]-RTI-55 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Potency of inhibiting 10 pM [125I]-RTI-55 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibitory activity against dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 83nMAssay Description:Potency of inhibiting [3H]WIN-35428 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Potency of inhibiting 10 pM [125I]-RTI-55 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 114nMAssay Description:Potency of inhibiting 10 pM [125I]-RTI-55 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 164nMAssay Description:Potency of inhibiting 10 pM [125I]-RTI-55 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 272nMAssay Description:Inhibitory activity against dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 446nMAssay Description:Inhibitory activity against dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 446nMAssay Description:Potency of inhibiting 10 pM [125I]RTI-55 binding to dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 465nMAssay Description:Inhibitory activity against dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 465nMAssay Description:Potency of inhibiting 10 pM [125I]RTI-55 binding to dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 637nMAssay Description:Inhibitory activity against dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 850nMAssay Description:Potency of inhibiting 10 pM [125I]RTI-55 binding to dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 850nMAssay Description:Inhibitory activity against dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Potency of inhibiting 10 pM [125I]-RTI-55 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 1.02E+3nMAssay Description:Potency of inhibiting 10 pM [125I]-RTI-55 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibitory activity against dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibitory activity against dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.93E+3nMAssay Description:Inhibitory activity against dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.05E+3nMAssay Description:Potency of inhibiting 10 pM [125I]RTI-55 binding to dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.05E+3nMAssay Description:Inhibitory activity against dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 2.08E+3nMAssay Description:Potency of inhibiting 10 pM [125I]-RTI-55 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 2.75E+3nMAssay Description:Potency of inhibiting 10 pM [125I]-RTI-55 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.16E+3nMAssay Description:Potency of inhibiting 10 pM [125I]RTI-55 binding to dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 6.47E+3nMAssay Description:Potency of inhibiting 10 pM [125I]-RTI-55 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rat)
State University of New York
Curated by ChEMBL
State University of New York
Curated by ChEMBL
Affinity DataIC50: 7.43E+3nMAssay Description:Potency of inhibiting 10 pM [125I]-RTI-55 binding to dopamine receptor in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Ability to displace 0.4 nM [3H]paroxetine binding to serotonin transporter in rat frontal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Ability to displace 0.4 nM [3H]paroxetine binding to serotonin transporter in rat frontal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Ability to displace 0.4 nM [3H]paroxetine binding to serotonin transporter in rat frontal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Ability to displace 0.4 nM [3H]paroxetine binding to serotonin transporter in rat frontal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Ability to displace 0.4 nM [3H]paroxetine binding to serotonin transporter in rat frontal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Ability to displace 0.4 nM [3H]paroxetine binding to serotonin transporter in rat frontal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 245nMAssay Description:Ability to displace 0.4 nM [3H]paroxetine binding to serotonin transporter in rat frontal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 245nMAssay Description:Ability to displace 0.4 nM [3H]paroxetine binding to serotonin transporter in rat frontal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 1.08E+3nMAssay Description:Ability to displace 0.4 nM [3H]paroxetine binding to serotonin transporter in rat frontal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Ability to displace 0.4 nM [3H]paroxetine binding to serotonin transporter in rat frontal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 2.02E+3nMAssay Description:Ability to displace 0.4 nM [3H]paroxetine binding to serotonin transporter in rat frontal cortexMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to displace 0.4 nM [3H]paroxetine binding to serotonin transporter in rat frontal cortexMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to displace 0.4 nM [3H]paroxetine binding to serotonin transporter in rat frontal cortexMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to displace 0.4 nM [3H]paroxetine binding to serotonin transporter in rat frontal cortexMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Ability to displace 0.4 nM [3H]paroxetine binding to serotonin transporter in rat frontal cortexMore data for this Ligand-Target Pair
