Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 5460
TargetNociceptin receptor(Human)
Purdue Pharma Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM86492(CAS_170713-75-4 | NSC_6324645 | Nociceptin)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Purdue Pharma Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM86491([8-(3,3-Diphenyl-propyl)-4-oxo-1-phenyl-1,3,8-tria...)
Affinity DataKi:  0.760nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Purdue Pharma Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM86258(CAS_23552-18-3 | NSC_5980 | Morphine)
Affinity DataKi:  2.06nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMu-type opioid receptor(Human)
Purdue Pharma Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM86493(CAS_27943 | NALTREXONE-HCl | NSC_27943 | Naltrexon...)
Affinity DataKi:  2.39nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Purdue Pharma Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM21130(U69,593 | N-methyl-N-(7-(1-pyrrolidinyl)-1-oxaspir...)
Affinity DataKi:  3.69nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Purdue Pharma Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM86258(CAS_23552-18-3 | NSC_5980 | Morphine)
Affinity DataKi:  134nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Purdue Pharma Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM86491([8-(3,3-Diphenyl-propyl)-4-oxo-1-phenyl-1,3,8-tria...)
Affinity DataKi:  243nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2012
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Purdue Pharma Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM86491([8-(3,3-Diphenyl-propyl)-4-oxo-1-phenyl-1,3,8-tria...)
Affinity DataKi:  286nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Purdue Pharma Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM86260(Naloxone(-) | NSC_10064 | CAS_465-65-6 | NALOXONE)
Affinity DataKi:  488nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Purdue Pharma Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM86258(CAS_23552-18-3 | NSC_5980 | Morphine)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2012
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Purdue Pharma Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM86258(CAS_23552-18-3 | NSC_5980 | Morphine)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2012
Entry Details Article
PubMed