Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50037253
TargetE3 ubiquitin-protein ligase XIAP(Human)
University of Michigan Comprehensive Cancer Center

Curated by ChEMBL
LigandPNGBDBM50145767(AVPIAQKSEK-FAM | CHEMBL404788)
Affinity DataKd:  240nMAssay Description:Dissociation constant towards X-linked inhibitor of apoptosis (XIAP) BIR3 protein was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
University of Michigan Comprehensive Cancer Center

Curated by ChEMBL
LigandPNGBDBM50145768(AVPIAQKSEK | CHEMBL414396)
Affinity DataKd:  240nMAssay Description:Dissociation constant for XIAP BIR3 proteinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
University of Michigan Comprehensive Cancer Center

Curated by ChEMBL
LigandPNGBDBM50145770(6-Amino-2-[(S)-2-((S)-2-{(S)-2-[((R)-{1-[(S)-2-((S...)
Affinity DataKd:  38nMAssay Description:Dissociation constant for XIAP BIR3 protein in FP-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
University of Michigan Comprehensive Cancer Center

Curated by ChEMBL
LigandPNGBDBM50145772(ARPFAQK-FAM | CHEMBL384327)
Affinity DataKd:  38nMAssay Description:Dissociation constant towards X-linked inhibitor of apoptosis (XIAP) BIR3 protein was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
University of Michigan Comprehensive Cancer Center

Curated by ChEMBL
LigandPNGBDBM50145770(6-Amino-2-[(S)-2-((S)-2-{(S)-2-[((R)-{1-[(S)-2-((S...)
Affinity DataKd:  20nMAssay Description:Dissociation constant for XIAP BIR3 protein using different binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
University of Michigan Comprehensive Cancer Center

Curated by ChEMBL
LigandPNGBDBM50145771(ARPFAQK-FAM | CHEMBL441156)
Affinity DataIC50: 570nMAssay Description:Compound was tested for inhibitory activity towards XIAP BIR3 proteinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
University of Michigan Comprehensive Cancer Center

Curated by ChEMBL
LigandPNGBDBM50145770(6-Amino-2-[(S)-2-((S)-2-{(S)-2-[((R)-{1-[(S)-2-((S...)
Affinity DataIC50: 570nMAssay Description:Inhibitory concentration of compound against XIAP BIR3 proteinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
University of Michigan Comprehensive Cancer Center

Curated by ChEMBL
LigandPNGBDBM50145767(AVPIAQKSEK-FAM | CHEMBL404788)
Affinity DataIC50: 2.80E+3nMAssay Description:Compound was tested for inhibitory activity towards XIAP BIR3 proteinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
University of Michigan Comprehensive Cancer Center

Curated by ChEMBL
LigandPNGBDBM50145768(AVPIAQKSEK | CHEMBL414396)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibitory concentration of compound against XIAP BIR3 proteinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
University of Michigan Comprehensive Cancer Center

Curated by ChEMBL
LigandPNGBDBM50145767(AVPIAQKSEK-FAM | CHEMBL404788)
Affinity DataIC50: 2.83E+3nMAssay Description:Compound was tested for inhibitory activity towards XIAP BIR3 proteinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
University of Michigan Comprehensive Cancer Center

Curated by ChEMBL
LigandPNGBDBM50145768(AVPIAQKSEK | CHEMBL414396)
Affinity DataIC50: 2.83E+3nMAssay Description:Inhibitory concentration of compound against XIAP BIR3 proteinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
University of Michigan Comprehensive Cancer Center

Curated by ChEMBL
LigandPNGBDBM13158(2,5-dihydroxy-3-undecylcyclohexa-2,5-diene-1,4-dio...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibitory concentration of compound against XIAP BIR3 proteinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
University of Michigan Comprehensive Cancer Center

Curated by ChEMBL
LigandPNGBDBM13158(2,5-dihydroxy-3-undecylcyclohexa-2,5-diene-1,4-dio...)
Affinity DataIC50: 4.10E+3nMAssay Description:Compound was tested for inhibitory activity towards XIAP BIR3 proteinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed