Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 4251
TargetG1/S-specific cyclin-D1(Human)
Cyclacel

LigandPNGBDBM59097(Aminopyrimidine, 10)
Affinity DataIC50: 7nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Cyclacel

LigandPNGBDBM59088(PD0183812)
Affinity DataIC50: 8nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM6619(3-[(9bR)-5-oxo-1H,2H,3H,5H,9bH-benzo[a]pyrrolizin-...)
Affinity DataIC50: 96nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-D1(Human)
Cyclacel

LigandPNGBDBM59092(Aminopyrimidine, 2)
Affinity DataIC50: 110nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-D1(Human)
Cyclacel

LigandPNGBDBM59095(Aminopyrimidine, 7)
Affinity DataIC50: 160nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM59088(PD0183812)
Affinity DataIC50: 165nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Cyclacel

LigandPNGBDBM59089(NSC625987)
Affinity DataIC50: 200nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Cyclacel

LigandPNGBDBM59090(Pyrazol-3-yl urea)
Affinity DataIC50: 200nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Cyclacel

LigandPNGBDBM59097(Aminopyrimidine, 10)
Affinity DataIC50: 220nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-D1(Human)
Cyclacel

LigandPNGBDBM59091(Aminopyrimidine, 1)
Affinity DataIC50: 230nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Cyclacel

LigandPNGBDBM50319624(Aminopyrimidine, 4 | CHEMBL1084454 | N1-(4-(2,4-Di...)
Affinity DataIC50: 230nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Cyclacel

LigandPNGBDBM59092(Aminopyrimidine, 2)
Affinity DataIC50: 330nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Cyclacel

LigandPNGBDBM59087(CHEMBL258765 | Fascaplysin | Fasca-plysi)
Affinity DataIC50: 350nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Cyclacel

LigandPNGBDBM59091(Aminopyrimidine, 1)
Affinity DataIC50: 410nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Cyclacel

LigandPNGBDBM59093(Aminopyrimidine, 3)
Affinity DataIC50: 430nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-D1(Human)
Cyclacel

LigandPNGBDBM59096(Aminopyrimidine, 8)
Affinity DataIC50: 430nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-D1(Human)
Cyclacel

LigandPNGBDBM59094(Aminopyrimidine, 6)
Affinity DataIC50: 640nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-D1(Human)
Cyclacel

LigandPNGBDBM59093(Aminopyrimidine, 3)
Affinity DataIC50: 890nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Cyclacel

LigandPNGBDBM50277583(2-amino-4-methyl-1,3-thiazol-5-yl)-N-[4-(morpholin...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Cyclacel

LigandPNGBDBM59095(Aminopyrimidine, 7)
Affinity DataIC50: 1.02E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Cyclacel

LigandPNGBDBM59094(Aminopyrimidine, 6)
Affinity DataIC50: 1.10E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Cyclacel

LigandPNGBDBM50319619(Aminopyrimidine, 5 | CHEMBL1085626 | 4-(2,4-Dimeth...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Cyclacel

LigandPNGBDBM59096(Aminopyrimidine, 8)
Affinity DataIC50: 2.20E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-D1(Human)
Cyclacel

LigandPNGBDBM50277583(2-amino-4-methyl-1,3-thiazol-5-yl)-N-[4-(morpholin...)
Affinity DataIC50: 2.40E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-D1(Human)
Cyclacel

LigandPNGBDBM50319624(Aminopyrimidine, 4 | CHEMBL1084454 | N1-(4-(2,4-Di...)
Affinity DataIC50: 3.80E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetG1/S-specific cyclin-D1(Human)
Cyclacel

LigandPNGBDBM50319619(Aminopyrimidine, 5 | CHEMBL1085626 | 4-(2,4-Dimeth...)
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM59090(Pyrazol-3-yl urea)
Affinity DataIC50: 2.50E+4nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM59087(CHEMBL258765 | Fascaplysin | Fasca-plysi)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM59089(NSC625987)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2011
Entry Details Article
PubMed