Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50035402
TargetGlutathione hydrolase 1 proenzyme(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50148335(1-Carboxy-3-[2-(carboxymethyl-carbamoyl)-ethanesul...)
Affinity DataKi:  5.30E+4nMpH: 8.0Assay Description:Compound tested for the inhibition of Gamma-glutamyltranspeptidase in rat kidney at pH 8.0 at 37 degree C (Competitive inhibition)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
TargetGlutathione hydrolase 1 proenzyme(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50148333((S)-1-Carboxy-3-[4-(carboxymethyl-carbamoyl)-pheny...)
Affinity DataKi:  2.30E+5nMpH: 8.0Assay Description:Compound tested for the inhibition of Gamma-glutamyltranspeptidase in rat kidney at pH 8.0 at 37 degree C (Competitive inhibition)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
TargetGlutathione hydrolase 1 proenzyme(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50148336((1S)-1-carboxy-3-({2-[(carboxymethyl)amino]-2-oxoe...)
Affinity DataKi:  5.20E+5nMpH: 8.0Assay Description:Compound tested for the inhibition of Gamma-glutamyltranspeptidase in rat kidney at pH 8.0 at 37 degree C (Competitive inhibition)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
TargetGlutathione hydrolase 1 proenzyme(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50148332(1-Carboxy-3-[2-(carboxymethyl-carbamoyl)-ethanesul...)
Affinity DataKi:  3.50E+6nMpH: 8.0Assay Description:Compound tested for the inhibition of Gamma-glutamyltranspeptidase in rat kidney at pH 8.0 at 37 degree CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
TargetGlutathione hydrolase 1 proenzyme(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50142500(L-methionine | (2S)-2-amino-4-(methylsulfanyl)buta...)
Affinity DataKi:  2.69E+7nMpH: 8.0Assay Description:Compound tested for the inhibition of Gamma-glutamyltranspeptidase in rat kidney at pH 8.0 at 37 degree C (Competitive inhibition)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
TargetGlutathione hydrolase 1 proenzyme(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50366922(METHIONINE SULFOXIDE)
Affinity DataKi:  5.90E+6nMpH: 8.0Assay Description:Compound tested for the inhibition of Gamma-glutamyltranspeptidase in rat kidney at pH 8.0 at 37 degree C (Competitive inhibition)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed