Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50014990
TargetMelanin-concentrating hormone receptor 1(Human)
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150059(N-(4-methyl-2-(pyrrolidin-1-yl)quinolin-6-yl)-2-(4...)
Affinity DataIC50: 10nMAssay Description:Tested for MCH-1 induced [Ca2+] release from CHO cells transfected with human MCH-1RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150063(N-[4-Methyl-2-(4-methyl-piperazin-1-yl)-quinolin-6...)
Affinity DataIC50: 63nMAssay Description:Tested for MCH-1 induced [Ca2+] release from CHO cells transfected with human MCH-1RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150057(2-(4-Chloro-phenoxy)-N-[4-methyl-2-(4-methyl-piper...)
Affinity DataIC50: 71nMAssay Description:Tested for MCH-1 induced [Ca2+] release from CHO cells transfected with human MCH-1RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150064(N-(4-Methyl-2-morpholin-4-yl-quinolin-6-yl)-2-(4-t...)
Affinity DataIC50: 124nMAssay Description:Tested for MCH-1 induced [Ca2+] release from CHO cells transfected with human MCH-1RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150072(2-(2,3-Dichloro-phenoxy)-N-[4-methyl-2-(4-methyl-p...)
Affinity DataIC50: 201nMAssay Description:Inhibitory activity against human 5-HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150057(2-(4-Chloro-phenoxy)-N-[4-methyl-2-(4-methyl-piper...)
Affinity DataIC50: 349nMAssay Description:Inhibitory activity against human 5-HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150061(N-(2-Isopropylamino-4-methyl-quinolin-6-yl)-2-(4-t...)
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against human 5-HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150063(N-[4-Methyl-2-(4-methyl-piperazin-1-yl)-quinolin-6...)
Affinity DataIC50: 442nMAssay Description:Inhibitory activity against human 5-HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150057(2-(4-Chloro-phenoxy)-N-[4-methyl-2-(4-methyl-piper...)
Affinity DataIC50: 970nMAssay Description:Inhibitory activity against human 5-HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150057(2-(4-Chloro-phenoxy)-N-[4-methyl-2-(4-methyl-piper...)
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibitory activity against human 5-HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed