Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50015136
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151871(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 0.300nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151874(Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-Met) | CHEMBL362...)
Affinity DataIC50: 0.300nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151880(YSTCYFIM | CHEMBL426697)
Affinity DataIC50: 1nMAssay Description:Concentration required to antagonise accessory gene regulator C3 of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151876(GVNACSSLF | CHEMBL182783)
Affinity DataIC50: 1nMAssay Description:Concentration required to antagonise accessory gene regulator C3 of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151873(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 2.80nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151876(GVNACSSLF | CHEMBL182783)
Affinity DataIC50: 2.90nMAssay Description:Antagonistic concentration for accessory gene regulator C1 of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151876(GVNACSSLF | CHEMBL182783)
Affinity DataEC50:  3.60nMAssay Description:Effective concentration to antagonise accessory gene regulator C2 of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151880(YSTCYFIM | CHEMBL426697)
Affinity DataIC50: 4nMAssay Description:Concentration required to antagonise accessory gene regulator C2 of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151877(N-[9-Benzyl-6-sec-butyl-12-methyl-3-(2-methylsulfa...)
Affinity DataIC50: 5nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151877(N-[9-Benzyl-6-sec-butyl-12-methyl-3-(2-methylsulfa...)
Affinity DataIC50: 5nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151879(2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylamino)...)
Affinity DataIC50: 6nMAssay Description:Concentration required to antagonise accessory gene regulator C2 of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151874(Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-Met) | CHEMBL362...)
Affinity DataIC50: 8nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151871(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 10nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151871(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 10nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151880(YSTCYFIM | CHEMBL426697)
Affinity DataEC50:  13nMAssay Description:Effective concentration to antagonise accessory gene regulator C4 of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151883(N-[9-Benzyl-6-sec-butyl-12-methyl-3-(2-methylsulfa...)
Affinity DataIC50: 19nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151874(Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-Met) | CHEMBL362...)
Affinity DataIC50: 21nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151874(Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-Met) | CHEMBL362...)
Affinity DataIC50: 21nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151879(2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylamino)...)
Affinity DataEC50:  26nMAssay Description:Effective concentration to antagonise accessory gene regulator C3 of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151879(2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylamino)...)
Affinity DataIC50: 70nMAssay Description:Antagonistic concentration for accessory gene regulator C1 of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151876(GVNACSSLF | CHEMBL182783)
Affinity DataIC50: 86nMAssay Description:Concentration required to antagonise accessory gene regulator C4 of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151873(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 137nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151879(2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylamino)...)
Affinity DataIC50: 150nMAssay Description:Concentration required to antagonise accessory gene regulator C4 of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151871(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 230nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151878(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 256nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151878(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50: 256nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151883(N-[9-Benzyl-6-sec-butyl-12-methyl-3-(2-methylsulfa...)
Affinity DataIC50: 295nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151872(2-{2-[4-(4-Benzoyl-phenoxy)-butyrylamino]-3-hydrox...)
Affinity DataIC50: 303nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151872(2-{2-[4-(4-Benzoyl-phenoxy)-butyrylamino]-3-hydrox...)
Affinity DataIC50: 303nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151875(N-(3-Benzyl-9,12-bis-hydroxymethyl-6-isobutyl-2,5,...)
Affinity DataIC50: 4.00E+3nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151875(N-(3-Benzyl-9,12-bis-hydroxymethyl-6-isobutyl-2,5,...)
Affinity DataIC50: 4.00E+3nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151880(YSTCYFIM | CHEMBL426697)
Affinity DataIC50: 7.00E+3nMAssay Description:Antagonistic concentration for accessory gene regulator C1 of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151881(Cyclo(Ac-Cys-Asp-Phe-Ile-Met) | CHEMBL362839)
Affinity DataIC50: 8.00E+3nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151882([15-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataEC50:  1.10E+4nMAssay Description:Effective concentration to antagonise accessory gene regulator C1 of Staphylococcus aureus; range = 9-11 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed