Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50015151
TargetTryptase beta-2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152197(2-[3-(5-Aminomethyl-2,4-dimethyl-benzylamino)-5-ch...)
Affinity DataKi:  93nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152198(2-[3-(4-Amino-cyclohexylamino)-5-chloro-6-methyl-2...)
Affinity DataKi:  138nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM16127(CHEMBL542712 | AIDS007118 | 2,2 -methanediylbis(1H...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152202(2-[3-(4-Amino-benzylamino)-5-chloro-6-methyl-2-oxo...)
Affinity DataKi:  245nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152200(N-(3-Aminomethyl-phenyl)-2-{5-chloro-6-methyl-2-ox...)
Affinity DataKi:  290nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152205(2-[3-(3-Aminomethyl-benzylamino)-5-chloro-6-methyl...)
Affinity DataKi:  390nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152206(N-(3-Aminomethyl-phenyl)-2-{5-chloro-3-[2-(1H-imid...)
Affinity DataKi:  426nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152196(N-(3-Aminomethyl-phenyl)-2-{5-chloro-6-methyl-2-ox...)
Affinity DataKi:  518nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152193(N-(3-Aminomethyl-phenyl)-2-{3-[(6-amino-2-methyl-p...)
Affinity DataKi:  580nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152203(2-[3-(4-Aminomethyl-benzylamino)-5-chloro-6-methyl...)
Affinity DataKi:  615nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152194(2-[3-(2-Amino-benzylamino)-5-chloro-6-methyl-2-oxo...)
Affinity DataKi:  875nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152204(N-(3-Aminomethyl-phenyl)-2-[5-chloro-3-(indan-2-yl...)
Affinity DataKi:  970nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152195(N-(3-Aminomethyl-phenyl)-2-[3-(4-benzoimidazol-1-y...)
Affinity DataKi:  1.24E+3nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152199(N-(3-Aminomethyl-phenyl)-2-(5-chloro-6-methyl-2-ox...)
Affinity DataKi:  1.55E+3nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2(Human)
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152201(N-(3-Aminomethyl-phenyl)-2-[5-chloro-3-(4-methoxy-...)
Affinity DataKi:  1.55E+3nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed