Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50015371
TargetSodium-dependent serotonin transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155461(3-(4-Iodo-phenyl)-8-aza-bicyclo[3.2.1]octane-2-car...)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155459(3-(4-Bromo-phenyl)-8-aza-bicyclo[3.2.1]octane-2-ca...)
Affinity DataKi:  0.240nMAssay Description:Displacement of [3H]cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50035766(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155452(3-(4-Bromo-phenyl)-8-aza-bicyclo[3.2.1]octane-2-ca...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155454(3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155457(3-(4-Bromo-phenyl)-8-aza-bicyclo[3.2.1]octane-2-ca...)
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155459(3-(4-Bromo-phenyl)-8-aza-bicyclo[3.2.1]octane-2-ca...)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H]CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155454(3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi:  0.620nMAssay Description:Displacement of [3H]cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155452(3-(4-Bromo-phenyl)-8-aza-bicyclo[3.2.1]octane-2-ca...)
Affinity DataKi:  0.720nMAssay Description:Displacement of [3H]CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155461(3-(4-Iodo-phenyl)-8-aza-bicyclo[3.2.1]octane-2-car...)
Affinity DataKi:  0.850nMAssay Description:Displacement of [3H]CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50106856(3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi:  0.930nMAssay Description:Displacement of [3H]CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155457(3-(4-Bromo-phenyl)-8-aza-bicyclo[3.2.1]octane-2-ca...)
Affinity DataKi:  0.950nMAssay Description:Displacement of [3H]cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155457(3-(4-Bromo-phenyl)-8-aza-bicyclo[3.2.1]octane-2-ca...)
Affinity DataKi:  1.02nMAssay Description:Displacement of [3H]-nisoxetine from norepinephrine transporter of rat cerebral corticex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155456(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  1.23nMAssay Description:Displacement of [3H]CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155456(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  1.65nMAssay Description:Displacement of [3H]cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155460(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  1.91nMAssay Description:Displacement of [3H]CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155451(3-(4-Bromo-phenyl)-8-(3-fluoro-propyl)-8-aza-bicyc...)
Affinity DataKi:  2.03nMAssay Description:Displacement of [3H]-nisoxetine from norepinephrine transporter of rat cerebral corticex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155453(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  2.33nMAssay Description:Displacement of [3H]CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155460(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  2.86nMAssay Description:Displacement of [3H]cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50106855(3-(4-Bromo-phenyl)-8-(3-fluoro-propyl)-8-aza-bicyc...)
Affinity DataKi:  3.33nMAssay Description:Displacement of [3H]CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50106856(3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi:  4.02nMAssay Description:Displacement of [3H]cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50035766(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  4.95nMAssay Description:Displacement of [3H]cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155460(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  5nMAssay Description:Inhibition of [18F]PET binding to dopamine transporter of human brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155459(3-(4-Bromo-phenyl)-8-aza-bicyclo[3.2.1]octane-2-ca...)
Affinity DataKi:  5nMAssay Description:Inhibition of [18F]PET binding to dopamine transporter of human brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155461(3-(4-Iodo-phenyl)-8-aza-bicyclo[3.2.1]octane-2-car...)
Affinity DataKi:  5nMAssay Description:Inhibition of [18F]PET binding to dopamine transporter of human brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155453(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  5nMAssay Description:Inhibition of [18F]PET binding to dopamine transporter of human brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155452(3-(4-Bromo-phenyl)-8-aza-bicyclo[3.2.1]octane-2-ca...)
Affinity DataKi:  5nMAssay Description:Inhibition of [18F]PET binding to dopamine transporter of human brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155453(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155452(3-(4-Bromo-phenyl)-8-aza-bicyclo[3.2.1]octane-2-ca...)
Affinity DataKi:  8.85nMAssay Description:Displacement of [3H]-nisoxetine from norepinephrine transporter of rat cerebral corticex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155451(3-(4-Bromo-phenyl)-8-(3-fluoro-propyl)-8-aza-bicyc...)
Affinity DataKi:  10.6nMAssay Description:Displacement of [3H]CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155459(3-(4-Bromo-phenyl)-8-aza-bicyclo[3.2.1]octane-2-ca...)
Affinity DataKi:  15.2nMAssay Description:Displacement of [3H]-nisoxetine from norepinephrine transporter of rat cerebral corticex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50035766(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  15.3nMAssay Description:Displacement of [3H]-nisoxetine from norepinephrine transporter of rat cerebral corticex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155451(3-(4-Bromo-phenyl)-8-(3-fluoro-propyl)-8-aza-bicyc...)
Affinity DataKi:  18.3nMAssay Description:Displacement of [3H]cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155458(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  25.7nMAssay Description:Displacement of [3H]CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155455(3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi:  30.8nMAssay Description:Displacement of [3H]cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50106855(3-(4-Bromo-phenyl)-8-(3-fluoro-propyl)-8-aza-bicyc...)
Affinity DataKi:  36.4nMAssay Description:Displacement of [3H]cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155458(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  38.7nMAssay Description:Displacement of [3H]cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155455(3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi:  44.5nMAssay Description:Displacement of [3H]CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50106856(3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]-nisoxetine from norepinephrine transporter of rat cerebral corticex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50106855(3-(4-Bromo-phenyl)-8-(3-fluoro-propyl)-8-aza-bicyc...)
Affinity DataKi:  196nMAssay Description:Displacement of [3H]-nisoxetine from norepinephrine transporter of rat cerebral corticex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155456(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  225nMAssay Description:Displacement of [3H]-nisoxetine from norepinephrine transporter of rat cerebral corticex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155460(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  244nMAssay Description:Displacement of [3H]-nisoxetine from norepinephrine transporter of rat cerebral corticex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155453(3-(4-Bromo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]-nisoxetine from norepinephrine transporter of rat cerebral corticex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155454(3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi:  413nMAssay Description:Displacement of [3H]-nisoxetine from norepinephrine transporter of rat cerebral corticex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155455(3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-nisoxetine from norepinephrine transporter of rat cerebral corticex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed