Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50000412
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataKi:  0.700nMAssay Description:Inhibition of [3H]L-364718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005459(CHEMBL9485 | CR 1409 | 4-(3,4-Dichloro-benzoylamin...)
Affinity DataKi:  49nMAssay Description:Inhibition of [3H]L-364718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005456(CHEMBL9308 | 1-(4-Chloro-phenyl)-3-(3,3-diphenyl-a...)
Affinity DataKi:  90nMAssay Description:Inhibition of [3H]L-364718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005471(CHEMBL9220 | 1H-Indole-2-carboxylic acid (3-phenyl...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]L-364718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005450(CHEMBL422036 | 1-(4-Chloro-phenyl)-3-(3-pentyl-oct...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]L-364718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005453(CHEMBL266596 | 1H-Indole-2-carboxylic acid [3,3-bi...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]L-364718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005455(CHEMBL8779 | 1H-Indole-2-carboxylic acid (3,3-diph...)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]L-364718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005466(CHEMBL9500 | 1H-Indole-2-carboxylic acid (3,3-diph...)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]L-364718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005468(CHEMBL8893 | 3,4-Dichloro-N-(3,3-diphenyl-allyl)-b...)
Affinity DataKi:  400nMAssay Description:Inhibition of [3H]L-364718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005457(CHEMBL9538 | 1-(4-Chloro-phenyl)-3-(4,4-diphenyl-b...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]L-364718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005470(CHEMBL8949 | Naphthalene-2-carboxylic acid (3,3-di...)
Affinity DataKi:  450nMAssay Description:Inhibition of [3H]L-364718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005461(CHEMBL9510 | Quinoline-2-carboxylic acid (3,3-diph...)
Affinity DataKi:  470nMAssay Description:Displacement of [3H]L-364718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005469(CHEMBL9312 | 1-(3,3-Diphenyl-allyl)-3-m-tolyl-urea)
Affinity DataKi:  800nMAssay Description:Inhibition of [3H]L-364718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005462(CHEMBL9379 | Naphthalene-1-carboxylic acid (3,3-di...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of [3H]L-364718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005467(CHEMBL9444 | 1-(4-Chloro-phenyl)-3-(2-diphenylamin...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]L-364718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005449(CHEMBL9174 | Quinoline-3-carboxylic acid (3,3-diph...)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]L-364718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005465(CHEMBL268197 | 4-Chloro-N-(3,3-diphenyl-allyl)-ben...)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of [3H]L-364718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005454(CHEMBL9181 | Quinoline-4-carboxylic acid (3,3-diph...)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]L-364718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005452(CHEMBL267507 | 1H-Indole-2-carboxylic acid (4,4-di...)
Affinity DataKi: >2.00E+3nMAssay Description:Compound was evaluated for its ability to inhibit [3H]L-364718 binding Cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005460(CHEMBL416144 | 5,6-Dihydro-4H-pyrrolo[3,2,1-ij]qui...)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]L-364718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005451(CHEMBL268382 | 1H-Indole-2-carboxylic acid [3,3-bi...)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]L-364718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005464(CHEMBL275031 | 1-(4-Chloro-phenyl)-3-[2-(10,11-dih...)
Affinity DataKi: >4.00E+3nMAssay Description:Inhibition of [3H]L-364718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005458(CHEMBL275126 | 1-(4-Chloro-phenyl)-3-(3-phenyl-all...)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]L-364718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed