Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50037484
TargetType-2 angiotensin II receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50049189(butyl 3-(4-((2-ethyl-5,7-dimethyl-3H-imidazo[4,5-b...)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50282396(PD-123319 | (S)-1-(4-Dimethylamino-3-methyl-benzyl...)
Affinity DataIC50: 34nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50369183(L-163491 | CHEMBL290214)
Affinity DataIC50: 101nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM82258(NSC_3961 | CAS_114798-26-4 | Losartan)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156173(butyl 3-(4-((1H-imidazol-1-yl)methyl)phenyl)-5-iso...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156167(butyl (5-isobutylthien-2-yl)sulfonylcarbamate deri...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50049189(butyl 3-(4-((2-ethyl-5,7-dimethyl-3H-imidazo[4,5-b...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156172(butyl (5-isobutylthien-2-yl)sulfonylcarbamate deri...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156168(butyl (5-isobutylthien-2-yl)sulfonylcarbamate deri...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156174(butyl (5-isobutylthien-2-yl)sulfonylcarbamate deri...)
Affinity DataKi:  7.10nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156175(butyl (5-isobutylthien-2-yl)sulfonylcarbamate deri...)
Affinity DataKi:  70nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156170(butyl (5-isobutylthien-2-yl)sulfonylcarbamate deri...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156171(butyl (5-isobutylthien-2-yl)sulfonylcarbamate deri...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156166(butyl (5-isobutylthien-2-yl)sulfonylcarbamate deri...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-Ang II from pig uterus membrane angiotensin II type 2 (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed