Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50037486
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50156214(2-(3,4-Dimethoxy-phenyl)-2-isopropyl-5-[4-(2-pheno...)
Affinity DataIC50: 400nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influx in the presence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50156213(omega-Conotoxin | CHEMBL439485)
Affinity DataIC50: 500nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influx in the presence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50156213(omega-Conotoxin | CHEMBL439485)
Affinity DataIC50: 600nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50156214(2-(3,4-Dimethoxy-phenyl)-2-isopropyl-5-[4-(2-pheno...)
Affinity DataIC50: 700nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50156215(1-(4-Amino-piperidin-1-yl)-4,4-bis-(4-fluoro-pheny...)
Affinity DataIC50: 1.03E+3nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50156215(1-(4-Amino-piperidin-1-yl)-4,4-bis-(4-fluoro-pheny...)
Affinity DataIC50: 2.40E+3nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influx in the presence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50156216(4-Methyl-2-methylamino-pentanoic acid {1-[4,4-bis-...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50156212(2-(3,4-Dimethoxy-phenyl)-2-isopropyl-5-[1-(2-pheno...)
Affinity DataIC50: 3.10E+3nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influx in the presence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50156212(2-(3,4-Dimethoxy-phenyl)-2-isopropyl-5-[1-(2-pheno...)
Affinity DataIC50: 3.80E+3nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed