Compile Data Set for Download or QSAR
Report error Found 142 Enz. Inhib. hit(s) with all data for entry = 50015502
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50128669(4-(4-but-2-ynyloxyphenylsulfanyl)piperidine-4-carb...)
Affinity DataIC50: 2nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156714(1-(4-bromobenzyl)-4-(4-prop-2-ynyloxybenzenesulfon...)
Affinity DataIC50: 3nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50411313(CHEMBL2096853)
Affinity DataIC50: 4nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50411313(CHEMBL2096853)
Affinity DataIC50: 4nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156718(1-(4-bromobenzyl)-4-(4-butoxyphenylsulfonyl)-N-hyd...)
Affinity DataIC50: 5nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156714(1-(4-bromobenzyl)-4-(4-prop-2-ynyloxybenzenesulfon...)
Affinity DataIC50: 6nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156695(1-benzyl-N-hydroxy-4-(4-(prop-2-ynyloxy)phenylsulf...)
Affinity DataIC50: 7nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156718(1-(4-bromobenzyl)-4-(4-butoxyphenylsulfonyl)-N-hyd...)
Affinity DataIC50: 10nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50128669(4-(4-but-2-ynyloxyphenylsulfanyl)piperidine-4-carb...)
Affinity DataIC50: 10nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156713(2-(4-methoxybenzenesulfonyl)octanoic acid hydroxya...)
Affinity DataIC50: 12nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156708(2-[4-(2-butynyloxy)phenyl]sulfonyl}-2-isopropyl-N-...)
Affinity DataIC50: 17nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50411317(CHEMBL2096740)
Affinity DataIC50: 17nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50411314(CHEMBL2096852)
Affinity DataIC50: 18nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156695(1-benzyl-N-hydroxy-4-(4-(prop-2-ynyloxy)phenylsulf...)
Affinity DataIC50: 18nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156705(2-{[4-(2-butynyloxy)phenyl]sulfonyl}-2-cyclohexyl-...)
Affinity DataIC50: 26nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50411315(CHEMBL2096739)
Affinity DataIC50: 28nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50411316(CHEMBL2096738)
Affinity DataIC50: 30nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156726(2-{[4-(2-butynyloxy)phenyl]sulfonyl}-N-hydroxy-2-(...)
Affinity DataIC50: 39nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156722(4-(4-but-2-ynyloxybenzenesulfonyl)-1-(4-methoxyben...)
Affinity DataIC50: 40nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156725(1-benzyl-4-(4-but-2-ynyloxybenzenesulfonyl)piperdi...)
Affinity DataIC50: 47nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50411312(CHEMBL2096855)
Affinity DataIC50: 48nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156698(2-(4-(but-2-ynyloxy)phenylthio)-N-hydroxy-2-phenyl...)
Affinity DataIC50: 50nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156721(2-{[4-(2-butynyloxy)phenyl]sulfanyl}-N-hydroxy-2-(...)
Affinity DataIC50: 50nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156710(2-{[4-(2-butynyloxy)phenyl]sulfonyl}-N-hydroxy-2-t...)
Affinity DataIC50: 51nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156715(2-(4-(but-2-ynyloxy)phenylsulfonyl)-2-(1-(cyclopro...)
Affinity DataIC50: 54nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156717(4-(4-but-2-ynyloxybenzenesulfonyl)-1-(4-chlorobenz...)
Affinity DataIC50: 55nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156701(1-(4-bromobenzyl)-4-(4-but-2-ynyxoybenzenesulfonyl...)
Affinity DataIC50: 65nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156704(2-{[4-(2-butynyloxy)phenyl]sulfonyl}-2-phenyl-N-hy...)
Affinity DataIC50: 68nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156695(1-benzyl-N-hydroxy-4-(4-(prop-2-ynyloxy)phenylsulf...)
Affinity DataIC50: 69nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50411316(CHEMBL2096738)
Affinity DataIC50: 72nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50128669(4-(4-but-2-ynyloxyphenylsulfanyl)piperidine-4-carb...)
Affinity DataIC50: 72nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156718(1-(4-bromobenzyl)-4-(4-butoxyphenylsulfonyl)-N-hyd...)
Affinity DataIC50: 72nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50411318(CHEMBL2096854)
Affinity DataIC50: 74nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156716(2-(4-but-2-ynyloxybenzenelsulfonyl)octanoic acid h...)
Affinity DataIC50: 75nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156709(4-(4-but-2-ynyloxybenzenesulfonyl)-1-ethylpiperdin...)
Affinity DataIC50: 80nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156722(4-(4-but-2-ynyloxybenzenesulfonyl)-1-(4-methoxyben...)
Affinity DataIC50: 82nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156725(1-benzyl-4-(4-but-2-ynyloxybenzenesulfonyl)piperdi...)
Affinity DataIC50: 90nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156704(2-{[4-(2-butynyloxy)phenyl]sulfonyl}-2-phenyl-N-hy...)
Affinity DataIC50: 94nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156695(1-benzyl-N-hydroxy-4-(4-(prop-2-ynyloxy)phenylsulf...)
Affinity DataIC50: 96nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156714(1-(4-bromobenzyl)-4-(4-prop-2-ynyloxybenzenesulfon...)
Affinity DataIC50: 98nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156696(2-{[4-(2-butynyloxy)phenyl]sulfanyl}-2-cyclohexyl-...)
Affinity DataIC50: 105nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156727(2-(4-but-2-ynyloxyphenylsulfanyl)octanoic acid hyd...)
Affinity DataIC50: 105nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156708(2-[4-(2-butynyloxy)phenyl]sulfonyl}-2-isopropyl-N-...)
Affinity DataIC50: 107nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156720(2-{[4-(2-butynyloxy)phenyl]sulfonyl}-N-hydroxy-2-t...)
Affinity DataIC50: 113nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156713(2-(4-methoxybenzenesulfonyl)octanoic acid hydroxya...)
Affinity DataIC50: 119nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50156706(2-(1-acetyl-4-piperidinyl)-2-{[4-(2-butynyloxy)phe...)
Affinity DataIC50: 119nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156704(2-{[4-(2-butynyloxy)phenyl]sulfonyl}-2-phenyl-N-hy...)
Affinity DataIC50: 124nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156714(1-(4-bromobenzyl)-4-(4-prop-2-ynyloxybenzenesulfon...)
Affinity DataIC50: 143nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50411314(CHEMBL2096852)
Affinity DataIC50: 148nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156725(1-benzyl-4-(4-but-2-ynyloxybenzenesulfonyl)piperdi...)
Affinity DataIC50: 148nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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