Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50015564
TargetDelta-type opioid receptor(Rat)
University of Cagliary

Curated by ChEMBL
LigandPNGBDBM50157686(5-[({5-[(2S)-2-({2-[(2S)-2-amino-3-(4-hydroxy-2,6-...)
Affinity DataKi:  0.0350nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat brain synaptosomes P2 fractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliary

Curated by ChEMBL
LigandPNGBDBM50157684(H-Dmt-Tic-Glu-NH2 | CHEMBL2369958)
Affinity DataKi:  0.0600nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat brain synaptosomes P2 fractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliary

Curated by ChEMBL
LigandPNGBDBM50157684(H-Dmt-Tic-Glu-NH2 | CHEMBL2369958)
Affinity DataKi:  0.0600nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain synaptosomes P2 fractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliary

Curated by ChEMBL
LigandPNGBDBM50157685(H-Dmt-Tic-Glu-NH-(CH2)5-NH2 | CHEMBL225479)
Affinity DataKi:  0.220nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat brain synaptosomes P2 fractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliary

Curated by ChEMBL
LigandPNGBDBM50157684(H-Dmt-Tic-Glu-NH2 | CHEMBL2369958)
Affinity DataIC50: 2.60nMAssay Description:Agonistic activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked twitchMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliary

Curated by ChEMBL
LigandPNGBDBM50157686(5-[({5-[(2S)-2-({2-[(2S)-2-amino-3-(4-hydroxy-2,6-...)
Affinity DataKi:  152nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain synaptosomes P2 fractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliary

Curated by ChEMBL
LigandPNGBDBM50157685(H-Dmt-Tic-Glu-NH-(CH2)5-NH2 | CHEMBL225479)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain synaptosomes P2 fractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Cagliary

Curated by ChEMBL
LigandPNGBDBM50157684(H-Dmt-Tic-Glu-NH2 | CHEMBL2369958)
Affinity DataIC50: 1.00E+3nMAssay Description:Agonistic activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically evoked twitchMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Cagliary

Curated by ChEMBL
LigandPNGBDBM50157686(5-[({5-[(2S)-2-({2-[(2S)-2-amino-3-(4-hydroxy-2,6-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Agonistic activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically evoked twitchMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Cagliary

Curated by ChEMBL
LigandPNGBDBM50157685(H-Dmt-Tic-Glu-NH-(CH2)5-NH2 | CHEMBL225479)
Affinity DataIC50: 1.00E+3nMAssay Description:Agonistic activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically evoked twitchMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed