Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 1504
TargetRAC-alpha serine/threonine-protein kinase(Human)
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11819((3R,4R)-N-{4-[4-(2-hydroxy-5-piperidin-1-ylbenzoyl...)
Affinity DataIC50: 20nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2006
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11820(N-[(3R,4R)-4-[(4-{[5-(3,3-dimethylpiperidin-1-yl)-...)
Affinity DataIC50: 20nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2006
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11817((3R,4R)-N-{4-[4-(5-dimethylamino-2-hydroxybenzoyl)...)
Affinity DataIC50: 23nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2006
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bovine)
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11817((3R,4R)-N-{4-[4-(5-dimethylamino-2-hydroxybenzoyl)...)
Affinity DataIC50: 30nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2006
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11821(N-[(3R,4R)-4-[(4-{[5-(4,4-dimethylpiperidin-1-yl)-...)
Affinity DataIC50: 40nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2006
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bovine)
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11819((3R,4R)-N-{4-[4-(2-hydroxy-5-piperidin-1-ylbenzoyl...)
Affinity DataIC50: 400nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2006
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11818(N-[(3R,4R)-4-[(4-{[3-(3,3-dimethylpiperidin-2-yl)-...)
Affinity DataIC50: 750nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2006
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bovine)
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11821(N-[(3R,4R)-4-[(4-{[5-(4,4-dimethylpiperidin-1-yl)-...)
Affinity DataIC50: 1.70E+3nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2006
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bovine)
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11820(N-[(3R,4R)-4-[(4-{[5-(3,3-dimethylpiperidin-1-yl)-...)
Affinity DataIC50: 1.90E+3nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2006
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bovine)
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM11818(N-[(3R,4R)-4-[(4-{[3-(3,3-dimethylpiperidin-2-yl)-...)
Affinity DataIC50: 2.40E+3nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2006
Entry Details Article
PubMed