Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50015660
TargetKappa-type opioid receptor(Rat)
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50159165(2S,4aR,6a(R,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]U-69593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50159161((3S,4aS,4bR,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl...)
Affinity DataKi:  6nMAssay Description:Inhibition of [3H]U-69593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50159162((3S,4aR,4bS,6S,8R,8aR)-6-Acetoxy-3-furan-3-yl-4a,8...)
Affinity DataKi:  6nMAssay Description:Inhibition of [3H]U-69593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50159163(1-deoxosalvinorin | (3S,4aR,4bS,6R,8R,8aR,10aR)-6-...)
Affinity DataKi:  18nMAssay Description:Inhibition of [3H]U-69593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50159172((3S,4aR,4bS,6S,8R,8aR,10aR)-6-Formyloxy-3-furan-3-...)
Affinity DataKi:  18nMAssay Description:Inhibition of [3H]U-69593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50159173((3S,4aS,4bR,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl...)
Affinity DataKi:  59nMAssay Description:Inhibition of [3H]U-69593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50159168((2S,4aR,6aR,7R,9S,10aS,10bR)-methyl 9-acetoxy-6a,1...)
Affinity DataKi:  156nMAssay Description:Inhibition of [3H]U-69593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50159169(Salvinorin A (ester) | (3S,4aR,4bS,6S,8R,8aR,10aS)...)
Affinity DataKi:  163nMAssay Description:Inhibition of [3H]U-69593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50159170(Acetic acid (3S,4aR,4bS,6S,8R,8aS,10aR)-3-furan-3-...)
Affinity DataKi:  347nMAssay Description:Inhibition of [3H]U-69593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50159171((3S,4aR,4bR,5R,6S,8aR,10aR)-5,6-Diacetoxy-3-furan-...)
Affinity DataKi:  1.02E+3nMAssay Description:Inhibition of [3H]U-69593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50159166((3S,4aR,4bS,5R,6S,8R,8aR,10aR)-5,6-Diacetoxy-3-fur...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]U-69593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50159167((3S,4aR,4bR,5R,6S,8aR,10aR)-6-Acetoxy-3-furan-3-yl...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]diprenorphine binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50159174((3S,4aR,4bR,5R,6S,8aR,10aR)-5-Acetoxy-3-furan-3-yl...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]U-69593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed