Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 1684
LigandPNGBDBM13344(N-[4-Chloro-3-(3-pyridinyloxymethyl)phenyl]-3-fluo...)
Affinity DataIC50: 65nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13354(3-(3-tert-butyl-1-phenyl-1H-pyrazol-5-yl)-1-(4-chl...)
Affinity DataIC50: 196nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13336(4-{4-(4-fluorophenyl)-2-[4-(methylsulfinyl)phenyl]...)
Affinity DataIC50: 290nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13353(3-fluoro-5-(morpholin-4-yl)-N-{1-[2-(pyridin-4-yl)...)
Affinity DataIC50: 340nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM13345(3-(3-tert-butyl-1H-pyrazol-5-yl)-1-{4-chloro-3-[(p...)
Affinity DataIC50: 350nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13351(3-fluoro-5-morpholin-4-yl-N-[3-(2-pyridin-4-ylethy...)
Affinity DataIC50: 630nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13349(2-({4-[2-(1H-indol-3-yl)ethyl]pyrimidin-2-yl}amino...)
Affinity DataIC50: 1.50E+3nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13342(2-[5-(2,6-Dichlorobenzyloxy)-2-pyridinylamino]-2-m...)
Affinity DataIC50: 2.40E+4nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13343(N-[4-Chloro-3-(3-pyridinyloxymethyl)phenyl]benzami...)
Affinity DataIC50: 3.00E+4nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13346(3-(2-(4-Pyridyl)ethyl)indole | 3-[2-(pyridin-4-yl)...)
Affinity DataIC50: 3.50E+4nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13340(3-(naphthalen-1-ylmethoxy)pyridin-2-amine | 2-Amin...)
Affinity DataIC50: 4.40E+4nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM13339(2-Amino-3-(2,6-dichlorobenzyloxy)pyridine | 3-[(2,...)
Affinity DataIC50: 1.09E+5nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13348(3-[2-(2-chloropyrimidin-4-yl)ethyl]-1H-indole | In...)
Affinity DataIC50: 1.20E+5nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13350(3-fluoro-N-1H-indol-5-yl-5-morpholin-4-ylbenzamide...)
Affinity DataIC50: 1.62E+5nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13352(1-[2-(pyridin-4-yl)ethyl]-1H-indole | 1-(2-(4-Pyri...)
Affinity DataIC50: 1.85E+5nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13341(2-({5-[(2,6-dichlorophenyl)methoxy]pyridin-2-yl}am...)
Affinity DataIC50: 2.00E+5nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13347(3-[2-(pyrimidin-4-yl)ethyl]-1H-indole | 3-(2-pyrim...)
Affinity DataIC50: 7.20E+5nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13338(3-(benzyloxy)pyridine | Pyridine derived fragment ...)
Affinity DataIC50: 1.00E+6nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed
LigandPNGBDBM13337(3-(benzyloxy)pyridin-2-amine | Pyridine derived fr...)
Affinity DataIC50: 1.30E+6nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMedPDB3D3D Structure (crystal)