Compile Data Set for Download or QSAR
Report error Found 84 Enz. Inhib. hit(s) with all data for entry = 50041387
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20598(2-(3-hydroxyphenyl)-1-methyl-1-{4-[2-(pyrrolidin-1...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20599(2-(3-hydroxyphenyl)-1-methyl-1-{4-[2-(piperidin-1-...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20589(1-{4-[2-(azepan-1-yl)ethoxy]phenyl}-1-methyl-2-phe...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20592(2-(4-fluorophenyl)-1-methyl-1-{4-[2-(pyrrolidin-1-...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20587(1-methyl-2-phenyl-1-{4-[2-(pyrrolidin-1-yl)ethoxy]...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20593(2-(4-fluorophenyl)-1-methyl-1-{4-[2-(piperidin-1-y...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20588(1-methyl-2-phenyl-1-{4-[2-(piperidin-1-yl)ethoxy]p...)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20596(1-methyl-2-[4-(propan-2-yl)phenyl]-1-{4-[2-(pyrrol...)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20591(1-methyl-2-(4-methylphenyl)-1-{4-[2-(piperidin-1-y...)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20601(2-(3-chlorophenyl)-1-methyl-1-{4-[2-(pyrrolidin-1-...)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20600(2-(3-fluorophenyl)-1-methyl-1-{4-[2-(pyrrolidin-1-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20595(2-(4-chlorophenyl)-1-methyl-1-{4-[2-(piperidin-1-y...)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20594(2-(4-chlorophenyl)-1-methyl-1-{4-[2-(pyrrolidin-1-...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20590(1-methyl-2-(4-methylphenyl)-1-{4-[2-(pyrrolidin-1-...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20602(2-(3-chlorophenyl)-1-methyl-1-{4-[2-(piperidin-1-y...)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20597(1-methyl-1-{4-[2-(piperidin-1-yl)ethoxy]phenyl}-2-...)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20585(2-phenyl-1-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-1...)
Affinity DataIC50: 10.7nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20603(1-methyl-1-{4-[2-(piperidin-1-yl)ethoxy]phenyl}-2-...)
Affinity DataIC50: 16.1nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20586(2-phenyl-1-{4-[2-(piperidin-1-yl)ethoxy]phenyl}-1,...)
Affinity DataIC50: 16.5nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20604(2-[3-(dimethylamino)phenyl]-1-methyl-1-{4-[2-(pyrr...)
Affinity DataIC50: 19.0nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20586(2-phenyl-1-{4-[2-(piperidin-1-yl)ethoxy]phenyl}-1,...)
Affinity DataIC50: 19.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM50410088(CHEMBL434346)
Affinity DataIC50: 19.8nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20585(2-phenyl-1-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-1...)
Affinity DataIC50: 21.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20594(2-(4-chlorophenyl)-1-methyl-1-{4-[2-(pyrrolidin-1-...)
Affinity DataIC50: 27.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20591(1-methyl-2-(4-methylphenyl)-1-{4-[2-(piperidin-1-y...)
Affinity DataIC50: 28.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20588(1-methyl-2-phenyl-1-{4-[2-(piperidin-1-yl)ethoxy]p...)
Affinity DataIC50: 29.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20590(1-methyl-2-(4-methylphenyl)-1-{4-[2-(pyrrolidin-1-...)
Affinity DataIC50: 31.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20598(2-(3-hydroxyphenyl)-1-methyl-1-{4-[2-(pyrrolidin-1...)
Affinity DataIC50: 31.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20592(2-(4-fluorophenyl)-1-methyl-1-{4-[2-(pyrrolidin-1-...)
Affinity DataIC50: 31.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20598(2-(3-hydroxyphenyl)-1-methyl-1-{4-[2-(pyrrolidin-1...)
Affinity DataIC50: 33.0nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20599(2-(3-hydroxyphenyl)-1-methyl-1-{4-[2-(piperidin-1-...)
Affinity DataIC50: 34.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20595(2-(4-chlorophenyl)-1-methyl-1-{4-[2-(piperidin-1-y...)
Affinity DataIC50: 35.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20593(2-(4-fluorophenyl)-1-methyl-1-{4-[2-(piperidin-1-y...)
Affinity DataIC50: 38.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20600(2-(3-fluorophenyl)-1-methyl-1-{4-[2-(pyrrolidin-1-...)
Affinity DataIC50: 39.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20587(1-methyl-2-phenyl-1-{4-[2-(pyrrolidin-1-yl)ethoxy]...)
Affinity DataIC50: 39.8nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20596(1-methyl-2-[4-(propan-2-yl)phenyl]-1-{4-[2-(pyrrol...)
Affinity DataIC50: 44.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20603(1-methyl-1-{4-[2-(piperidin-1-yl)ethoxy]phenyl}-2-...)
Affinity DataIC50: 46.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20599(2-(3-hydroxyphenyl)-1-methyl-1-{4-[2-(piperidin-1-...)
Affinity DataIC50: 47.0nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20602(2-(3-chlorophenyl)-1-methyl-1-{4-[2-(piperidin-1-y...)
Affinity DataIC50: 49.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20589(1-{4-[2-(azepan-1-yl)ethoxy]phenyl}-1-methyl-2-phe...)
Affinity DataIC50: 56.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20601(2-(3-chlorophenyl)-1-methyl-1-{4-[2-(pyrrolidin-1-...)
Affinity DataIC50: 66.1nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20597(1-methyl-1-{4-[2-(piperidin-1-yl)ethoxy]phenyl}-2-...)
Affinity DataIC50: 71.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM50410088(CHEMBL434346)
Affinity DataIC50: 71.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20589(1-{4-[2-(azepan-1-yl)ethoxy]phenyl}-1-methyl-2-phe...)
Affinity DataIC50: 80.0nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20592(2-(4-fluorophenyl)-1-methyl-1-{4-[2-(pyrrolidin-1-...)
Affinity DataIC50: 82.0nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20587(1-methyl-2-phenyl-1-{4-[2-(pyrrolidin-1-yl)ethoxy]...)
Affinity DataIC50: 83.0nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20588(1-methyl-2-phenyl-1-{4-[2-(piperidin-1-yl)ethoxy]p...)
Affinity DataIC50: 83.0nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20593(2-(4-fluorophenyl)-1-methyl-1-{4-[2-(piperidin-1-y...)
Affinity DataIC50: 92.0nMAssay Description:Inhibition of transcriptional activation by human estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20604(2-[3-(dimethylamino)phenyl]-1-methyl-1-{4-[2-(pyrr...)
Affinity DataIC50: 94.0nMAssay Description:Inhibition of binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Calcutta

Curated by ChEMBL
LigandPNGBDBM20588(1-methyl-2-phenyl-1-{4-[2-(piperidin-1-yl)ethoxy]p...)
Affinity DataIC50: 104nMAssay Description:Inhibition of binding to human estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
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