Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 766
LigandPNGBDBM5874(N-[5-(Ethylsulfonyl)-2-methoxyphenyl]-5-(3-thien-3...)
Affinity DataIC50: 15nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5873(N-[5-(ethanesulfonyl)-2-methoxyphenyl]-5-[3-(thiop...)
Affinity DataIC50: 16nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5870(4-(2-{[5-(ethanesulfonyl)-2-methoxyphenyl]amino}-1...)
Affinity DataIC50: 18nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5875(N-[5-(ethanesulfonyl)-2-methoxyphenyl]-5-[3-(pyrid...)
Affinity DataIC50: 22nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5862(5-(3-Chlorophenyl)-N-[5-(ethylsulfonyl)-2-methoxyp...)
Affinity DataIC50: 22nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5859(N,N-diethyl-4-methoxy-3-[(5-phenyl-1,3-oxazol-2-yl...)
Affinity DataIC50: 23nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5878(N-[5-(Ethylsulfonyl)-2-methoxyphenyl]-5-[3-(1-meth...)
Affinity DataIC50: 25nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5871(N-[5-(ethanesulfonyl)-2-methoxyphenyl]-5-(3-ethylp...)
Affinity DataIC50: 29nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5864(N-[5-(ethanesulfonyl)-2-methoxyphenyl]-5-(3-methox...)
Affinity DataIC50: 36nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM11445(N-(cyclopropylmethyl)-4-methoxy-3-({5-[3-(pyridin-...)
Affinity DataIC50: 38nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5881(N-[5-(Ethylsulfonyl)-2-methoxyphenyl]-5-(2 -chloro...)
Affinity DataIC50: 39nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5860(N-[5-(Ethylsulfonyl)-2-methoxyphenyl]-5-phenyl-1,3...)
Affinity DataIC50: 50nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5869(5-(4-Cyanophenyl)-N-[5-(ethylsulfonyl)-2-methoxyph...)
Affinity DataIC50: 51nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5876(N-[5-(Ethylsulfonyl)-2-methoxyphenyl]-5-(3-pyridin...)
Affinity DataIC50: 76nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5877(N-[5-(ethanesulfonyl)-2-methoxyphenyl]-5-[3-(pyrid...)
Affinity DataIC50: 78nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5879(N-[5-(ethanesulfonyl)-2-methoxyphenyl]-5-(3-phenyl...)
Affinity DataIC50: 79nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5868(N-[5-(ethanesulfonyl)-2-methoxyphenyl]-5-(4-fluoro...)
Affinity DataIC50: 79nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5867(5-(4-chlorophenyl)-N-[5-(ethanesulfonyl)-2-methoxy...)
Affinity DataIC50: 81nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5866(N-[5-(ethanesulfonyl)-2-methoxyphenyl]-5-(4-methox...)
Affinity DataIC50: 87nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5880(N-[5-(ethanesulfonyl)-2-methoxyphenyl]-5-[3-(2-flu...)
Affinity DataIC50: 89nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5872(1-[3-(2-{[5-(Ethylsulfonyl)-2-methoxyphenyl]amino}...)
Affinity DataIC50: 91nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5865(5-(3-Fluorophenyl)-N-[5-(ethylsulfonyl)-2-methoxyp...)
Affinity DataIC50: 93nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5858(5-phenyl-N-(3,4,5-trimethoxyphenyl)-1,3-oxazol-2-a...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5856(N-(3,4-dimethoxyphenyl)-5-phenyl-1,3-oxazol-2-amin...)
Affinity DataIC50: 140nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5863(3-(2-{[5-(ethanesulfonyl)-2-methoxyphenyl]amino}-1...)
Affinity DataIC50: 141nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5857(N-(3,5-Dimethoxyphenyl)-5-phenyl-1,3-oxazol-2-amin...)
Affinity DataIC50: 170nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5861(5-(2-chlorophenyl)-N-[5-(ethanesulfonyl)-2-methoxy...)
Affinity DataIC50: 360nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5848(N-(2-methoxyphenyl)-5-phenyl-1,3-oxazol-2-amine | ...)
Affinity DataIC50: 380nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5851({3-[(5-phenyl-1,3-oxazol-2-yl)amino]phenyl}methano...)
Affinity DataIC50: 500nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5854(4-[(5-phenyl-1,3-oxazol-2-yl)amino]benzene-1-sulfo...)
Affinity DataIC50: 500nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5852(N-(3-(Ethylsulfonyl)phenyl)-5-phenyl-1,3-oxazol-2-...)
Affinity DataIC50: 720nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5847(N-(2-Cyanophenyl)-5-phenyl-1,3-oxazol-2-amine Hydr...)
Affinity DataIC50: 870nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5853(N-(3-Methylphenyl)-5-phenyl-1,3-oxazol-2-amine | 2...)
Affinity DataIC50: 870nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5849(3-[(5-phenyl-1,3-oxazol-2-yl)amino]benzonitrile | ...)
Affinity DataIC50: 930nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5364(N,5-diphenyl-1,3-oxazol-2-amine | 2-Anilino-5-aryl...)
Affinity DataIC50: 1.20E+3nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5850(N-(3-Phenoxyphenyl)-5-phenyl-1,3-oxazol-2-amine | ...)
Affinity DataIC50: 1.41E+3nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed
LigandPNGBDBM5855(N-(4-Phenoxyphenyl)-5-phenyl-1,3-oxazol-2-amine | ...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2005
Entry Details Article
PubMed