Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 5495
TargetMelanocortin receptor 4(Human)
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM82411(CAS_75921-69-6 | NDP-MSH)
Affinity DataKi:  3.98nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM86683(NBI-58702)
Affinity DataKi:  6.31nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM50152808(4-(2R)-[(3R)-1,2,3,4-tetrahydroisoquinolinylcarbox...)
Affinity DataKi:  9.55nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM50119368((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  10.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMelanocortin receptor 4(Human)
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM86681(NBI-58704)
Affinity DataKi:  13.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM86682(CAS_114843 | NSC_114843 | Beta MSH)
Affinity DataKi:  18.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM86684(NBI-56297)
Affinity DataKi:  20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM82406(desacetyl-alpha-MSH)
Affinity DataKi:  30.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM50152798(CHEMBL182231 | NBI-56453 | 1,2,3,4-Tetrahydro-isoq...)
Affinity DataKi:  74.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM82407(Gamma1-MSH)
Affinity DataKi:  589nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2012
Entry Details Article
PubMed