Compile Data Set for Download or QSAR
Report error Found 75 Enz. Inhib. hit(s) with all data for entry = 50015945
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162738(1-Benzoyl-4-(4-but-2-ynyloxy-benzenesulfonyl)-[1,4...)
Affinity DataIC50: 4nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162730(4-Acetyl-1-(4-but-2-ynyloxy-benzenesulfonyl)-[1,4]...)
Affinity DataIC50: 4nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162744(1-{[4-(but-2-yn-1-yloxy)benzene]sulfonyl}-N-hydrox...)
Affinity DataIC50: 5nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162742(4-(4-But-2-ynyloxy-benzenesulfonyl)-5-hydroxycarba...)
Affinity DataIC50: 5nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162731(1-Benzyl-4-(4-but-2-ynyloxy-benzenesulfonyl)-[1,4]...)
Affinity DataIC50: 7nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162735({2-[4-(4-But-2-ynyloxy-benzenesulfonyl)-3-hydroxyc...)
Affinity DataIC50: 7nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162740(4-(4-But-2-ynyloxy-benzenesulfonyl)-1,1-dioxo-1lam...)
Affinity DataIC50: 8nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162736(4-(4-But-2-ynyloxy-benzenesulfonyl)-1-isobutyryl-[...)
Affinity DataIC50: 9nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162729(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-(thiophene-2...)
Affinity DataIC50: 10nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162738(1-Benzoyl-4-(4-but-2-ynyloxy-benzenesulfonyl)-[1,4...)
Affinity DataIC50: 10nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162753(1-(4-But-2-ynyloxy-benzenesulfonyl)-[1,4]diazepane...)
Affinity DataIC50: 11nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162741(4-(4-But-2-ynyloxy-benzenesulfonyl)-[1,4]thiazepan...)
Affinity DataIC50: 11nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162728(4-(2-Amino-acetyl)-1-(4-but-2-ynyloxy-benzenesulfo...)
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162741(4-(4-But-2-ynyloxy-benzenesulfonyl)-[1,4]thiazepan...)
Affinity DataIC50: 13nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162754(4-(4-But-2-ynyloxy-benzenesulfonyl)-[1,4]diazepane...)
Affinity DataIC50: 14nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162745(4-(4-(but-2-ynyloxy)phenylsulfonyl)-N-hydroxy-1-(2...)
Affinity DataIC50: 15nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162739(4-(4-(but-2-ynyloxy)phenylsulfonyl)-1-ethyl-N-hydr...)
Affinity DataIC50: 17nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162743(4-Benzoyl-1-(4-but-2-ynyloxy-benzenesulfonyl)-[1,4...)
Affinity DataIC50: 17nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162740(4-(4-But-2-ynyloxy-benzenesulfonyl)-1,1-dioxo-1lam...)
Affinity DataIC50: 19nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162750(4-(4-But-2-ynyloxy-benzenesulfonyl)-1-propionyl-[1...)
Affinity DataIC50: 19nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162749(4-(4-But-2-ynyloxy-benzenesulfonyl)-[1,4]thiazepan...)
Affinity DataIC50: 20nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162750(4-(4-But-2-ynyloxy-benzenesulfonyl)-1-propionyl-[1...)
Affinity DataIC50: 20nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162733(4-(4-But-2-ynyloxy-benzenesulfonyl)-1-methyl-[1,4]...)
Affinity DataIC50: 21nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162733(4-(4-But-2-ynyloxy-benzenesulfonyl)-1-methyl-[1,4]...)
Affinity DataIC50: 23nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162736(4-(4-But-2-ynyloxy-benzenesulfonyl)-1-isobutyryl-[...)
Affinity DataIC50: 23nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162748(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-methyl-[1,4]...)
Affinity DataIC50: 24nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162746(4-(4-(but-2-ynyloxy)phenylsulfonyl)-N-hydroxy-1,4-...)
Affinity DataIC50: 24nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162734(4-(4-But-2-ynyloxy-benzenesulfonyl)-1,1-dioxo-1lam...)
Affinity DataIC50: 28nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162751(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-(propane-1-s...)
Affinity DataIC50: 30nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162745(4-(4-(but-2-ynyloxy)phenylsulfonyl)-N-hydroxy-1-(2...)
Affinity DataIC50: 31nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162746(4-(4-(but-2-ynyloxy)phenylsulfonyl)-N-hydroxy-1,4-...)
Affinity DataIC50: 32nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162747(4-(4-But-2-ynyloxy-benzenesulfonyl)-3-hydroxycarba...)
Affinity DataIC50: 35nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162749(4-(4-But-2-ynyloxy-benzenesulfonyl)-[1,4]thiazepan...)
Affinity DataIC50: 36nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162739(4-(4-(but-2-ynyloxy)phenylsulfonyl)-1-ethyl-N-hydr...)
Affinity DataIC50: 37nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162737(4-Benzyl-1-(4-but-2-ynyloxy-benzenesulfonyl)-[1,4]...)
Affinity DataIC50: 52nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162737(4-Benzyl-1-(4-but-2-ynyloxy-benzenesulfonyl)-[1,4]...)
Affinity DataIC50: 61nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162743(4-Benzoyl-1-(4-but-2-ynyloxy-benzenesulfonyl)-[1,4...)
Affinity DataIC50: 65nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162752(4-Benzenesulfonyl-1-(4-but-2-ynyloxy-benzenesulfon...)
Affinity DataIC50: 68nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162742(4-(4-But-2-ynyloxy-benzenesulfonyl)-5-hydroxycarba...)
Affinity DataIC50: 74nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162732(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-(4-dimethyla...)
Affinity DataIC50: 75nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50162731(1-Benzyl-4-(4-but-2-ynyloxy-benzenesulfonyl)-[1,4]...)
Affinity DataIC50: 83nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162752(4-Benzenesulfonyl-1-(4-but-2-ynyloxy-benzenesulfon...)
Affinity DataIC50: 88nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162742(4-(4-But-2-ynyloxy-benzenesulfonyl)-5-hydroxycarba...)
Affinity DataIC50: 92nMAssay Description:Inhibitory concentration against matrix metalloprotease-1 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162738(1-Benzoyl-4-(4-but-2-ynyloxy-benzenesulfonyl)-[1,4...)
Affinity DataIC50: 113nMAssay Description:Inhibitory concentration against matrix metalloprotease-1 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162740(4-(4-But-2-ynyloxy-benzenesulfonyl)-1,1-dioxo-1lam...)
Affinity DataIC50: 114nMAssay Description:Inhibitory concentration against matrix metalloprotease-1 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162744(1-{[4-(but-2-yn-1-yloxy)benzene]sulfonyl}-N-hydrox...)
Affinity DataIC50: 128nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162751(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-(propane-1-s...)
Affinity DataIC50: 140nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162729(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-(thiophene-2...)
Affinity DataIC50: 142nMAssay Description:Inhibitory concentration against Matrix metalloprotease-13 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162736(4-(4-But-2-ynyloxy-benzenesulfonyl)-1-isobutyryl-[...)
Affinity DataIC50: 142nMAssay Description:Inhibitory concentration against matrix metalloprotease-1 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162741(4-(4-But-2-ynyloxy-benzenesulfonyl)-[1,4]thiazepan...)
Affinity DataIC50: 171nMAssay Description:Inhibitory concentration against matrix metalloprotease-1 at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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