Compile Data Set for Download or QSAR
Report error Found 61 Enz. Inhib. hit(s) with all data for entry = 50016029
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163958([6-Chloro-3-(3-fluoro-phenyl)-5-(2-fluoro-phenyl)-...)
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163993([3-(3-Fluoro-phenyl)-5-(2-fluoro-phenyl)-4-oxo-3,4...)
Affinity DataIC50: 140nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163950([3-(3-Fluoro-phenyl)-5-(3-methoxy-phenyl)-4-oxo-3,...)
Affinity DataIC50: 140nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163988([3-(3-Fluoro-phenyl)-5-(2-methoxy-phenyl)-4-oxo-3,...)
Affinity DataIC50: 140nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163973([3-(3-Fluoro-phenyl)-5-(2-fluoro-phenyl)-6-methyl-...)
Affinity DataIC50: 150nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163983((6-Methyl-4-oxo-3,5-diphenyl-3,4-dihydro-thieno[2,...)
Affinity DataIC50: 160nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163970([3-(2-Fluoro-phenyl)-4-oxo-5-phenyl-3,4-dihydro-th...)
Affinity DataIC50: 160nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163964([3-(3-Fluoro-phenyl)-4-oxo-5-phenyl-3,4,5,6,7,8-he...)
Affinity DataIC50: 170nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163962([3-(3-Fluoro-phenyl)-4-oxo-5-phenyl-3,4-dihydro-th...)
Affinity DataIC50: 180nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163991([3-(3-Fluoro-phenyl)-5-methyl-4-oxo-3,4,5,6,7,8-he...)
Affinity DataIC50: 200nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163950([3-(3-Fluoro-phenyl)-5-(3-methoxy-phenyl)-4-oxo-3,...)
Affinity DataIC50: 210nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163947([3-(3-Fluoro-phenyl)-5-isopropyl-4-oxo-3,4-dihydro...)
Affinity DataIC50: 230nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163957((4-Oxo-3,5-diphenyl-3,4-dihydro-thieno[2,3-d]pyrim...)
Affinity DataIC50: 250nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163962([3-(3-Fluoro-phenyl)-4-oxo-5-phenyl-3,4-dihydro-th...)
Affinity DataIC50: 250nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163980([3-(3-Fluoro-phenyl)-5-(4-methoxy-phenyl)-4-oxo-3,...)
Affinity DataIC50: 280nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163981([3,5-Bis-(3-fluoro-phenyl)-4-oxo-3,4-dihydro-thien...)
Affinity DataIC50: 290nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163971([5-(4-Fluoro-phenyl)-4-oxo-3-phenyl-3,4-dihydro-th...)
Affinity DataIC50: 290nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163975([3-(4-Fluoro-phenyl)-4-oxo-5-phenyl-3,4-dihydro-th...)
Affinity DataIC50: 320nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163956([3-(3-Fluoro-phenyl)-4-oxo-3,4,5,6,7,8-hexahydro-b...)
Affinity DataIC50: 450nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163948([3-(3-Methoxy-phenyl)-4-oxo-5-phenyl-3,4-dihydro-t...)
Affinity DataIC50: 470nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163992((4-Oxo-5-phenyl-3-pyridin-3-yl-3,4-dihydro-thieno[...)
Affinity DataIC50: 480nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163970([3-(2-Fluoro-phenyl)-4-oxo-5-phenyl-3,4-dihydro-th...)
Affinity DataIC50: 500nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163994([3-(3-Fluoro-phenyl)-7-methyl-4-oxo-3,4,5,6,7,8-he...)
Affinity DataIC50: 530nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163971([5-(4-Fluoro-phenyl)-4-oxo-3-phenyl-3,4-dihydro-th...)
Affinity DataIC50: 800nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163957((4-Oxo-3,5-diphenyl-3,4-dihydro-thieno[2,3-d]pyrim...)
Affinity DataIC50: 800nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163948([3-(3-Methoxy-phenyl)-4-oxo-5-phenyl-3,4-dihydro-t...)
Affinity DataIC50: 820nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163966([3-(3-Fluoro-phenyl)-5-(2-fluoro-phenyl)-6-isoprop...)
Affinity DataIC50: 900nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163964([3-(3-Fluoro-phenyl)-4-oxo-5-phenyl-3,4,5,6,7,8-he...)
Affinity DataIC50: 930nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163989(3-(3-Fluoro-phenyl)-2-hydrazinocarbonylmethylsulfa...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163992((4-Oxo-5-phenyl-3-pyridin-3-yl-3,4-dihydro-thieno[...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163984(3-(6-Methyl-4-oxo-3,5-diphenyl-3,4-dihydro-thieno[...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163975([3-(4-Fluoro-phenyl)-4-oxo-5-phenyl-3,4-dihydro-th...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163951([3-(3-Fluoro-phenyl)-5-(2-hydroxy-phenyl)-4-oxo-3,...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163965([3-(3-Fluoro-phenyl)-4-oxo-6-phenyl-3,4-dihydro-qu...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163977([3-(3-Chloro-phenyl)-4-oxo-5-phenyl-3,4-dihydro-th...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163954([3-(2-Chloro-phenyl)-4-oxo-5-phenyl-3,4-dihydro-th...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163963([3-(4-Chloro-phenyl)-4-oxo-5-phenyl-3,4-dihydro-th...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163968([3-(2-Methoxy-phenyl)-4-oxo-5-phenyl-3,4-dihydro-t...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163953([3-(4-Methoxy-phenyl)-4-oxo-5-phenyl-3,4-dihydro-t...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163946([5-Benzyl-3-(3-fluoro-phenyl)-4-oxo-3,4,5,6,7,8-he...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163990((3-Benzyl-4-oxo-5-phenyl-3,4-dihydro-thieno[2,3-d]...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163985((3-Cyclohexyl-4-oxo-5-phenyl-3,4-dihydro-thieno[2,...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163959((4-Oxo-3,5-diphenyl-3,4-dihydro-thieno[2,3-d]pyrim...)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163949((4-Oxo-3,5-diphenyl-3,4-dihydro-thieno[2,3-d]pyrim...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163969([5-[2-(3-Diethylamino-propoxy)-phenyl]-3-(3-fluoro...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163972(2-(3-Amino-2-oxo-propylsulfanyl)-3-(3-fluoro-pheny...)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163945([3-(3-Fluoro-phenyl)-4-oxo-7-propyl-3,4,5,6,7,8-he...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163995([3-(4-Fluoro-phenyl)-5-methyl-4-oxo-3,4-dihydro-th...)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163982([3-(3-Fluoro-phenyl)-4-oxo-3,4,5,6,7,8-hexahydro-p...)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibitory concentration against tissue transglutaminase was determined using full progress curvesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50163987((3-Methyl-4-oxo-5-phenyl-3,4-dihydro-thieno[2,3-d]...)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibitory concentration against tissue transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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