Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50000468
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006122(CHEMBL49862 | 2-Benzyl-N-[1-(1-cyclohexylmethyl-2,...)
Affinity DataIC50: 0.360nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006125(CHEMBL297429 | 2-Benzyl-N-[1-(1-cyclohexylmethyl-2...)
Affinity DataIC50: 0.470nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006138(CHEMBL46607 | 2-(Morpholine-4-carbonyl)-3-phenyl-c...)
Affinity DataIC50: 0.700nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006123(CHEMBL296051 | 2,3-Diphenyl-cyclopropanecarboxylic...)
Affinity DataIC50: 1.10nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006128(CHEMBL431540 | 2-Isobutyl-3-(morpholine-4-carbonyl...)
Affinity DataIC50: 2.10nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006132(CHEMBL297929 | [1-[1-(1-Cyclohexylmethyl-2,3-dihyd...)
Affinity DataIC50: 2.40nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006122(CHEMBL49862 | 2-Benzyl-N-[1-(1-cyclohexylmethyl-2,...)
Affinity DataIC50: 8.30nMpH: 7.4Assay Description:In vitro potency against human plasma renin at pH 7.4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006124(CHEMBL301754 | 2-Ethyl-3-(morpholine-4-carbonyl)-c...)
Affinity DataIC50: 10nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006134(CHEMBL49460 | 2-Benzyl-3-(morpholine-4-carbonyl)-c...)
Affinity DataIC50: 10nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006119(CHEMBL46606 | 2-Ethyl-3-(morpholine-4-carbonyl)-cy...)
Affinity DataIC50: 16nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006127(CHEMBL49287 | 2-Isobutyl-3-(morpholine-4-carbonyl)...)
Affinity DataIC50: 19nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006138(CHEMBL46607 | 2-(Morpholine-4-carbonyl)-3-phenyl-c...)
Affinity DataIC50: 20nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006135(CHEMBL297928 | 2-Benzyl-3-(morpholine-4-carbonyl)-...)
Affinity DataIC50: 25nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006137(CHEMBL296028 | 2-Benzyl-3-(morpholine-4-carbonyl)-...)
Affinity DataIC50: 27nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006133(CHEMBL49541 | 2-Isobutyl-3-(morpholine-4-carbonyl)...)
Affinity DataIC50: 33nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006128(CHEMBL431540 | 2-Isobutyl-3-(morpholine-4-carbonyl...)
Affinity DataIC50: 41nMpH: 7.4Assay Description:In vitro potency against human plasma renin at pH 7.4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006139(CHEMBL295544 | 2-Isobutyl-3-(morpholine-4-carbonyl...)
Affinity DataIC50: 44nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006125(CHEMBL297429 | 2-Benzyl-N-[1-(1-cyclohexylmethyl-2...)
Affinity DataIC50: 54nMpH: 7.4Assay Description:In vitro potency against human plasma renin at pH 7.4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006120(CHEMBL298708 | 2-Ethyl-3-(morpholine-4-carbonyl)-c...)
Affinity DataIC50: 92nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006136(CHEMBL45604 | 2-(Morpholine-4-carbonyl)-3-phenyl-c...)
Affinity DataIC50: 120nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006121(CHEMBL296790 | 2-(Morpholine-4-carbonyl)-3-phenyl-...)
Affinity DataIC50: 120nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006129(CHEMBL296702 | 2-Benzyl-3-(morpholine-4-carbonyl)-...)
Affinity DataIC50: 120nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006130(CHEMBL47597 | 2-Benzyl-N-[1-(1-cyclohexylmethyl-2,...)
Affinity DataIC50: 150nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006131(CHEMBL299824 | 2-(Morpholine-4-carbonyl)-3-phenyl-...)
Affinity DataIC50: 200nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006126(CHEMBL298277 | 2-Ethyl-3-(morpholine-4-carbonyl)-c...)
Affinity DataIC50: 200nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006124(CHEMBL301754 | 2-Ethyl-3-(morpholine-4-carbonyl)-c...)
Affinity DataIC50: 230nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006132(CHEMBL297929 | [1-[1-(1-Cyclohexylmethyl-2,3-dihyd...)
Affinity DataIC50: 300nMpH: 7.4Assay Description:In vitro potency against human plasma renin at pH 7.4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006134(CHEMBL49460 | 2-Benzyl-3-(morpholine-4-carbonyl)-c...)
Affinity DataIC50: 370nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006119(CHEMBL46606 | 2-Ethyl-3-(morpholine-4-carbonyl)-cy...)
Affinity DataIC50: 610nMpH: 6.0Assay Description:In vitro inhibition of purified human renin at a pH of 6.0.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006123(CHEMBL296051 | 2,3-Diphenyl-cyclopropanecarboxylic...)
Affinity DataIC50: 810nMpH: 7.4Assay Description:In vitro potency against human plasma renin at pH 7.4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006135(CHEMBL297928 | 2-Benzyl-3-(morpholine-4-carbonyl)-...)
Affinity DataIC50: 1.00E+3nMpH: 7.4Assay Description:In vitro potency against human plasma renin at pH 7.4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRenin(Human)
University of Texas

Curated by ChEMBL
LigandPNGBDBM50006127(CHEMBL49287 | 2-Isobutyl-3-(morpholine-4-carbonyl)...)
Affinity DataIC50: 1.00E+3nMpH: 7.4Assay Description:In vitro potency against human plasma renin at pH 7.4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed