Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50034537
TargetVascular endothelial growth factor receptor 2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50363958(CHEMBL1952211)
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant EE-tagged intracellular domain of KDR using biotin-EEEEYFELVAKKKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50363957(CHEMBL1952210)
Affinity DataIC50: 44nMAssay Description:Inhibition of human recombinant EE-tagged intracellular domain of KDR using biotin-EEEEYFELVAKKKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50363957(CHEMBL1952210)
Affinity DataIC50: 44nMAssay Description:Inhibition of human recombinant EE-tagged intracellular domain of KDR using biotin-EEEEYFELVAKKKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50363957(CHEMBL1952210)
Affinity DataIC50: 310nMAssay Description:Inhibition of human recombinant His-tagged intracellular domain of EGFR using biotin-EEEEYFELV as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50363957(CHEMBL1952210)
Affinity DataIC50: 310nMAssay Description:Inhibition of human recombinant His-tagged intracellular domain of EGFR using biotin-EEEEYFELV as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Fyn(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50363957(CHEMBL1952210)
Affinity DataIC50: 322nMAssay Description:Inhibition of Fyn by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50363958(CHEMBL1952211)
Affinity DataIC50: 365nMAssay Description:Inhibition of human recombinant His-tagged intracellular domain of EGFR using biotin-EEEEYFELV as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetEphrin type-B receptor 3(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50363957(CHEMBL1952210)
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of EphB3More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50363957(CHEMBL1952210)
Affinity DataIC50: 3.04E+3nMAssay Description:Inhibition of ERK2 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50363957(CHEMBL1952210)
Affinity DataIC50: 1.25E+5nMAssay Description:Inhibition of PKCalpha by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Sgk1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50363957(CHEMBL1952210)
Affinity DataIC50: 1.25E+5nMAssay Description:Inhibition of SGKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50363957(CHEMBL1952210)
Affinity DataIC50: 1.25E+5nMAssay Description:Inhibition of PKCdelta by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50363957(CHEMBL1952210)
Affinity DataIC50: 1.25E+5nMAssay Description:Inhibition of CDK1/cyclin B by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed