Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50016461
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169328(5-{4-[3-(5-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-...)
Affinity DataKi:  1.10nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169314(2-Furan-2-yl-7-pyridin-2-yl-[1,2,4]triazolo[1,5-c]...)
Affinity DataKi:  1.40nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169318(2-Furan-2-yl-7-pyridin-4-yl-[1,2,4]triazolo[1,5-c]...)
Affinity DataKi:  1.90nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169326(7-(3-{4-[3,5-Difluoro-4-(2-methoxy-ethoxy)-phenyl]...)
Affinity DataKi:  2.20nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169313(2-Furan-2-yl-7-[3-(4-thiazol-2-yl-piperazin-1-ylme...)
Affinity DataKi:  2.40nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169331(2-Furan-2-yl-7-(3-{4-[4-(2-methoxy-ethoxy)-2-methy...)
Affinity DataKi:  2.70nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169312(7-(3-{4-[2-Fluoro-4-(2-methoxy-ethoxy)-phenyl]-pip...)
Affinity DataKi:  2.70nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169323(2-Furan-2-yl-7-(3-{4-[4-(2-methoxy-ethoxy)-phenyl]...)
Affinity DataKi:  2.80nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169317([3-(5-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyr...)
Affinity DataKi:  2.80nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169309(7-(2,4-Dimethoxy-phenyl)-2-furan-2-yl-[1,2,4]triaz...)
Affinity DataKi:  2.90nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169332(7-(3-{4-[2-Chloro-4-(2-methoxy-ethoxy)-phenyl]-pip...)
Affinity DataKi:  2.90nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169304(2-Furan-2-yl-7-(3-{4-[3-methoxy-4-(2-methoxy-ethox...)
Affinity DataKi:  3.30nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169306(2-{4-[3-(5-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-...)
Affinity DataKi:  3.60nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169339(2-Furan-2-yl-7-{3-[(methyl-phenethyl-amino)-methyl...)
Affinity DataKi:  3.60nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169322(2-Furan-2-yl-7-m-tolyl-[1,2,4]triazolo[1,5-c]pyrim...)
Affinity DataKi:  3.70nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169324(2-Furan-2-yl-7-(3-{4-[3-(2-methoxy-ethoxy)-phenyl]...)
Affinity DataKi:  4nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169338(2-(furan-2-yl)-7-(2-methoxyphenyl)-[1,2,4]triazolo...)
Affinity DataKi:  4.30nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169315(2-Furan-2-yl-7-thiophen-2-yl-[1,2,4]triazolo[1,5-c...)
Affinity DataKi:  4.40nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169333(2-Furan-2-yl-7-(2,3,4-trimethoxy-phenyl)-[1,2,4]tr...)
Affinity DataKi:  4.5nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169319(7-(2,5-Dimethoxy-phenyl)-2-furan-2-yl-[1,2,4]triaz...)
Affinity DataKi:  4.5nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169330(2-Furan-2-yl-7-(3,4,5-trimethoxy-phenyl)-[1,2,4]tr...)
Affinity DataKi:  4.5nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169321(2-Furan-2-yl-7-[3-(4-phenyl-piperidin-1-ylmethyl)-...)
Affinity DataKi:  4.60nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169316(2-Furan-2-yl-7-[3-(4-phenyl-piperazin-1-ylmethyl)-...)
Affinity DataKi:  4.60nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169336(2-Furan-2-yl-7-(4-isopropyl-phenyl)-[1,2,4]triazol...)
Affinity DataKi:  4.70nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169301(7-(3-Amino-phenyl)-2-furan-2-yl-[1,2,4]triazolo[1,...)
Affinity DataKi:  5nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169334(2-Furan-2-yl-7-(3-methoxy-phenyl)-[1,2,4]triazolo[...)
Affinity DataKi:  5nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169310(3-(5-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyri...)
Affinity DataKi:  5.40nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169303(7-Biphenyl-3-yl-2-furan-2-yl-[1,2,4]triazolo[1,5-c...)
Affinity DataKi:  5.5nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169335(7-(3-{4-[2,6-Difluoro-4-(2-methoxy-ethoxy)-phenyl]...)
Affinity DataKi:  6.40nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169300(2-Furan-2-yl-7-pyridin-3-yl-[1,2,4]triazolo[1,5-c]...)
Affinity DataKi:  6.60nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169307(2-Furan-2-yl-7-phenyl-[1,2,4]triazolo[1,5-c]pyrimi...)
Affinity DataKi:  7nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169308(7-(3,4-Dimethoxy-phenyl)-2-furan-2-yl-[1,2,4]triaz...)
Affinity DataKi:  7.30nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169305(2-Furan-2-yl-7-(4-methoxy-phenyl)-[1,2,4]triazolo[...)
Affinity DataKi:  7.30nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169320(7-{3-[4-(4-Fluoro-phenyl)-piperidin-1-ylmethyl]-ph...)
Affinity DataKi:  7.40nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169327(2-Furan-2-yl-7-p-tolyl-[1,2,4]triazolo[1,5-c]pyrim...)
Affinity DataKi:  8.40nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169337(2-Furan-2-yl-7-(3-{4-[4-(2-methoxy-ethoxy)-phenyl]...)
Affinity DataKi:  8.90nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169325(7-{3-[4-(3,4-Dichloro-phenyl)-piperazin-1-ylmethyl...)
Affinity DataKi:  11nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169311(2-Furan-2-yl-7-o-tolyl-[1,2,4]triazolo[1,5-c]pyrim...)
Affinity DataKi:  22nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169302(7-(2,3-Dimethoxy-phenyl)-2-furan-2-yl-[1,2,4]triaz...)
Affinity DataKi:  22nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169329(7-(2,6-Dimethoxy-phenyl)-2-furan-2-yl-[1,2,4]triaz...)
Affinity DataKi:  1.70E+3nMAssay Description:In vitro ability to displace [3H]SCH-58261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed