Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50016531
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50065796(2-[2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-quino...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in strand transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50065796(2-[2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-quino...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in standard 3'-processing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170145({2-[(E)-2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-...)
Affinity DataIC50: 7.00E+4nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in strand transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170146({2-[(E)-2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in standard 3'-processing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170146({2-[(E)-2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in strand transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170145({2-[(E)-2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in standard 3'-processing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170149((3,4-Difluoro-phenyl)-{2-[(E)-2-(3,4-dihydroxy-phe...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in strand transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170144({2-[(E)-2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in strand transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170144({2-[(E)-2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in standard 3'-processing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170148({2-[(E)-2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in standard 3'-processing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170148({2-[(E)-2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in strand transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170149((3,4-Difluoro-phenyl)-{2-[(E)-2-(3,4-dihydroxy-phe...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in standard 3'-processing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed