Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50016547
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170333(JWH-302 | 2-(3-methoxyphenyl)-1-(1-pentyl-1H-indol...)
Affinity DataEC50:  24.4nMAssay Description:Effective concentration for stimulation of [35S]GTP-gamma-S, binding at CB2 receptor in presence of 3 uM CP-55940More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170339(JWH-251 | 1-(1-pentyl-1H-indol-3-yl)-2-o-tolyletha...)
Affinity DataEC50:  29nMAssay Description:Effective concentration for stimulation of [35S]GTP-gamma-S binding at CB1 receptor in presence of 10 uM WIN-55212-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170333(JWH-302 | 2-(3-methoxyphenyl)-1-(1-pentyl-1H-indol...)
Affinity DataEC50:  29.3nMAssay Description:Effective concentration for stimulation of [35S]GTP-gamma-S binding at CB1 receptor in presence of 10 uM WIN-55212-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170339(JWH-251 | 1-(1-pentyl-1H-indol-3-yl)-2-o-tolyletha...)
Affinity DataEC50:  8.30nMAssay Description:Effective concentration for stimulation of [35S]GTP-gamma-S, binding at CB2 receptor in presence of 3 uM CP-55940More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataKi:  0.280nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170357(JWH-203 | 2-(2-Chloro-phenyl)-1-(1-pentyl-1H-indol...)
Affinity DataKi:  7nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170357(JWH-203 | 2-(2-Chloro-phenyl)-1-(1-pentyl-1H-indol...)
Affinity DataKi:  8nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170337(2-(2-bromophenyl)-1-(1-pentyl-1H-indol-3-yl)ethano...)
Affinity DataKi:  8.40nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170335(2-(2-Methoxy-phenyl)-1-(1-pentyl-1H-indol-3-yl)-et...)
Affinity DataKi:  11nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170356(2-(2-chlorophenyl)-1-(2-methyl-1-pentyl-1H-indol-3...)
Affinity DataKi:  13nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170345(JWH-305 | 2-(2-bromophenyl)-1-(2-methyl-1-pentyl-1...)
Affinity DataKi:  15nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170333(JWH-302 | 2-(3-methoxyphenyl)-1-(1-pentyl-1H-indol...)
Affinity DataKi:  17nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170343(1-(2-Methyl-1-pentyl-1H-indol-3-yl)-2-o-tolyl-etha...)
Affinity DataKi:  19nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170337(2-(2-bromophenyl)-1-(1-pentyl-1H-indol-3-yl)ethano...)
Affinity DataKi:  20nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170343(1-(2-Methyl-1-pentyl-1H-indol-3-yl)-2-o-tolyl-etha...)
Affinity DataKi:  23nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170331(2-(2-Fluoro-phenyl)-1-(1-pentyl-1H-indol-3-yl)-eth...)
Affinity DataKi:  23nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170356(2-(2-chlorophenyl)-1-(2-methyl-1-pentyl-1H-indol-3...)
Affinity DataKi:  25nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170342(JWH-306 | 2-(2-Methoxy-phenyl)-1-(2-methyl-1-penty...)
Affinity DataKi:  25nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170345(JWH-305 | 2-(2-bromophenyl)-1-(2-methyl-1-pentyl-1...)
Affinity DataKi:  29nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170339(JWH-251 | 1-(1-pentyl-1H-indol-3-yl)-2-o-tolyletha...)
Affinity DataKi:  29nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170335(2-(2-Methoxy-phenyl)-1-(1-pentyl-1H-indol-3-yl)-et...)
Affinity DataKi:  33nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  36nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170332(JWH-237 | 2-(3-Chloro-phenyl)-1-(1-pentyl-1H-indol...)
Affinity DataKi:  38nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170354(JWH-314 | 2-(2-fluorophenyl)-1-(2-methyl-1-pentyl-...)
Affinity DataKi:  39nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170331(2-(2-Fluoro-phenyl)-1-(1-pentyl-1H-indol-3-yl)-eth...)
Affinity DataKi:  39nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  41nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170334(JWH-253 | 2-(3-methoxyphenyl)-1-(2-methyl-1-pentyl...)
Affinity DataKi:  62nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170344(2-(3-Fluoro-phenyl)-1-(1-pentyl-1H-indol-3-yl)-eth...)
Affinity DataKi:  72nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170354(JWH-314 | 2-(2-fluorophenyl)-1-(2-methyl-1-pentyl-...)
Affinity DataKi:  76nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170342(JWH-306 | 2-(2-Methoxy-phenyl)-1-(2-methyl-1-penty...)
Affinity DataKi:  82nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170334(JWH-253 | 2-(3-methoxyphenyl)-1-(2-methyl-1-pentyl...)
Affinity DataKi:  84nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170333(JWH-302 | 2-(3-methoxyphenyl)-1-(1-pentyl-1H-indol...)
Affinity DataKi:  89nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170338(1-(1-pentyl-1H-indol-3-yl)-2-phenylethanone | 1-(1...)
Affinity DataKi:  90nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170344(2-(3-Fluoro-phenyl)-1-(1-pentyl-1H-indol-3-yl)-eth...)
Affinity DataKi:  91nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170332(JWH-237 | 2-(3-Chloro-phenyl)-1-(1-pentyl-1H-indol...)
Affinity DataKi:  106nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170355(JWH-303 | 2-(3-chlorophenyl)-1-(2-methyl-1-pentyl-...)
Affinity DataKi:  117nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170341(1-(2-Methyl-1-pentyl-1H-indol-3-yl)-2-phenyl-ethan...)
Affinity DataKi:  124nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170355(JWH-303 | 2-(3-chlorophenyl)-1-(2-methyl-1-pentyl-...)
Affinity DataKi:  138nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170339(JWH-251 | 1-(1-pentyl-1H-indol-3-yl)-2-o-tolyletha...)
Affinity DataKi:  146nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170338(1-(1-pentyl-1H-indol-3-yl)-2-phenylethanone | 1-(1...)
Affinity DataKi:  159nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170351(1-(1-Pentyl-1H-indol-3-yl)-2-p-tolyl-ethanone | JW...)
Affinity DataKi:  179nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170341(1-(2-Methyl-1-pentyl-1H-indol-3-yl)-2-phenyl-ethan...)
Affinity DataKi:  180nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170336(JWH-315 | 2-(3-Fluoro-phenyl)-1-(2-methyl-1-pentyl...)
Affinity DataKi:  182nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170330(2-(4-fluorophenyl)-1-(1-pentyl-1H-indol-3-yl)ethan...)
Affinity DataKi:  365nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170348(JWH-206 | 2-(4-chlorophenyl)-1-(1-pentyl-1H-indol-...)
Affinity DataKi:  389nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170330(2-(4-fluorophenyl)-1-(1-pentyl-1H-indol-3-yl)ethan...)
Affinity DataKi:  422nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170336(JWH-315 | 2-(3-Fluoro-phenyl)-1-(2-methyl-1-pentyl...)
Affinity DataKi:  430nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170353(JWH-201 | 2-(4-Methoxy-phenyl)-1-(1-pentyl-1H-indo...)
Affinity DataKi:  444nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170348(JWH-206 | 2-(4-chlorophenyl)-1-(1-pentyl-1H-indol-...)
Affinity DataKi:  498nMAssay Description:Binding affinity to displace [3H]CP-55940 from cloned human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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