Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50016654
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50050517(N-alkyl Gly-boro-Pro derivative | Boronic acid der...)
Affinity DataIC50: 0.300nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171653(N-alkyl Gly-boro-Pro derivative | CHEMBL196120)
Affinity DataIC50: 0.800nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171648(N-alkyl Gly-boro-Pro derivative | CHEMBL372180)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171649(N-alkyl Gly-boro-Pro derivative | CHEMBL196933)
Affinity DataIC50: 1.80nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171645(2-Cyclodecylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50: 2.20nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171650(2-Cyclooctonylamino-1-pyrrolidin-1-yl--2-borandihy...)
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171656(2-Cyclohexylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50: 4.10nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171647(N-alkyl Gly-boro-Pro derivative | CHEMBL373269)
Affinity DataIC50: 4.60nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171653(N-alkyl Gly-boro-Pro derivative | CHEMBL196120)
Affinity DataIC50: 6.30nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171649(N-alkyl Gly-boro-Pro derivative | CHEMBL196933)
Affinity DataIC50: 7.80nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171647(N-alkyl Gly-boro-Pro derivative | CHEMBL373269)
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171657(2-(Bicyclo[3.2.1]oct-6-ylamino)-1-((S)-2-dihydroxy...)
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50050517(N-alkyl Gly-boro-Pro derivative | Boronic acid der...)
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171644(N-alkyl Gly-boro-Pro derivative | CHEMBL427012)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171651(2-Cyclopentylamino-1-pyrrolidin-1-yl--2-borandihyd...)
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171651(2-Cyclopentylamino-1-pyrrolidin-1-yl--2-borandihyd...)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171657(2-(Bicyclo[3.2.1]oct-6-ylamino)-1-((S)-2-dihydroxy...)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171656(2-Cyclohexylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50: 27nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171650(2-Cyclooctonylamino-1-pyrrolidin-1-yl--2-borandihy...)
Affinity DataIC50: 27nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171652(N-alkyl Gly-boro-Pro derivative | CHEMBL381444)
Affinity DataIC50: 35nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50050517(N-alkyl Gly-boro-Pro derivative | Boronic acid der...)
Affinity DataIC50: 38nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171645(2-Cyclodecylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50: 58nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171648(N-alkyl Gly-boro-Pro derivative | CHEMBL372180)
Affinity DataIC50: 61nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171655(2-Cyclobutylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50: 75nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171644(N-alkyl Gly-boro-Pro derivative | CHEMBL427012)
Affinity DataIC50: 99nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171644(N-alkyl Gly-boro-Pro derivative | CHEMBL427012)
Affinity DataIC50: 120nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171658(2-Cyclopropylamino-1-pyrrolidin-1-yl--2-borandihyd...)
Affinity DataIC50: 130nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171655(2-Cyclobutylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50: 140nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171649(N-alkyl Gly-boro-Pro derivative | CHEMBL196933)
Affinity DataIC50: 150nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171657(2-(Bicyclo[3.2.1]oct-6-ylamino)-1-((S)-2-dihydroxy...)
Affinity DataIC50: 180nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171648(N-alkyl Gly-boro-Pro derivative | CHEMBL372180)
Affinity DataIC50: 270nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171650(2-Cyclooctonylamino-1-pyrrolidin-1-yl--2-borandihy...)
Affinity DataIC50: 290nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171647(N-alkyl Gly-boro-Pro derivative | CHEMBL373269)
Affinity DataIC50: 420nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171645(2-Cyclodecylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50: 530nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171652(N-alkyl Gly-boro-Pro derivative | CHEMBL381444)
Affinity DataIC50: 560nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171658(2-Cyclopropylamino-1-pyrrolidin-1-yl--2-borandihyd...)
Affinity DataIC50: 570nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171656(2-Cyclohexylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50: 650nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171652(N-alkyl Gly-boro-Pro derivative | CHEMBL381444)
Affinity DataIC50: 770nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171646(N-alkyl Gly-boro-Pro derivative | CHEMBL196188)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171646(N-alkyl Gly-boro-Pro derivative | CHEMBL196188)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171651(2-Cyclopentylamino-1-pyrrolidin-1-yl--2-borandihyd...)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171653(N-alkyl Gly-boro-Pro derivative | CHEMBL196120)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171654(N-alkyl Gly-boro-Pro derivative | CHEMBL434184)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171655(2-Cyclobutylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171646(N-alkyl Gly-boro-Pro derivative | CHEMBL196188)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed