Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50003735
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50223597(CHEMBL95777)
Affinity DataIC50: 1.82E+4nMAssay Description:Inhibitory activity against supercoiling activity of DNA gyrase isolated from Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50223617(CHEMBL95778)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibitory activity against supercoiling activity of DNA gyrase isolated from Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 4 subunit A(Escherichia coli (strain K12))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50223597(CHEMBL95777)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibitory activity against decatenation of DNA topoisomerase IV isolated from Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50475386(CHEMBL194702)
Affinity DataIC50: 3.26E+4nMAssay Description:Inhibitory activity against supercoiling activity of DNA gyrase isolated from Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 4 subunit A(Escherichia coli (strain K12))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50223617(CHEMBL95778)
Affinity DataIC50: 3.54E+4nMAssay Description:Inhibitory activity against decatenation of DNA topoisomerase IV isolated from Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 4 subunit A(Escherichia coli (strain K12))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50475386(CHEMBL194702)
Affinity DataIC50: 6.53E+4nMAssay Description:Inhibitory activity against decatenation of DNA topoisomerase IV isolated from Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed