Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50016871
TargetLeukotriene B4 receptor 1(Human)
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174609((LTB4-(Csa)4)2-Glu-H Conjugate | CHEMBL412510)
Affinity DataIC50: 8nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer, for 1 h at 37 degree ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174608(HYNIC Conjugate | CHEMBL406432)
Affinity DataIC50: 16nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 hr at 37 de...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174610(2-[5-Methyl-5-(1H-tetrazol-5-yl)-hexyloxy]-4,6-dip...)
Affinity DataIC50: 20nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer, for 1 hr at 37 degree...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174607(DTPA Conjugate | CHEMBL415548)
Affinity DataIC50: 30nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 hr at 37 de...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174606(HYNIC Analogue | CHEMBL384950)
Affinity DataIC50: 44nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 hr at 37 de...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174606(HYNIC Analogue | CHEMBL384950)
Affinity DataIC50: 45nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer upon incubation for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174607(DTPA Conjugate | CHEMBL415548)
Affinity DataIC50: 54nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer, for 1 h at 37 degree ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174611(HYNIC Conjugate | CHEMBL437275)
Affinity DataIC50: 230nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 hr at 37 de...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed